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In Vitro and In Vivo Evaluation of ABCG2 (BCRP) Inhibitors Derived from Ko143.
J Med Chem. 2023 May 25;66(10):6782-6797. doi: 10.1021/acs.jmedchem.3c00168. Epub 2023 May 8.
J Med Chem. 2023.
PMID: 37154765
Synthesis and Structure-Affinity Relationship of Small Molecules for Imaging Human CD80 by Positron Emission Tomography.
Taddio MF, Mu L, Castro Jaramillo CA, Bollmann T, Schmid DM, Muskalla LP, Gruene T, Chiotellis A, Ametamey SM, Schibli R, Krämer SD.
Taddio MF, et al.
J Med Chem. 2019 Sep 12;62(17):8090-8100. doi: 10.1021/acs.jmedchem.9b00858. Epub 2019 Aug 29.
J Med Chem. 2019.
PMID: 31430137
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Multi-parameter optimization: Development of a morpholin-3-one derivative with an improved kinetic profile for imaging monoacylglycerol lipase in the brain.
He Y, Grether U, Taddio MF, Meier C, Keller C, Edelmann MR, Honer M, Huber S, Wittwer MB, Heer D, Richter H, Collin L, Hug MN, Hilbert M, Postmus AGJ, Stevens AF, van der Stelt M, Krämer SD, Schibli R, Mu L, Gobbi LC.
He Y, et al. Among authors: taddio mf.
Eur J Med Chem. 2022 Dec 5;243:114750. doi: 10.1016/j.ejmech.2022.114750. Epub 2022 Sep 9.
Eur J Med Chem. 2022.
PMID: 36137365
Free article.
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Physiologically Based Pharmacokinetic Modelling with Dynamic PET Data to Study the In Vivo Effects of Transporter Inhibition on Hepatobiliary Clearance in Mice.
Taddio MF, Mu L, Keller C, Schibli R, Krämer SD.
Taddio MF, et al.
Contrast Media Mol Imaging. 2018 Jun 3;2018:5849047. doi: 10.1155/2018/5849047. eCollection 2018.
Contrast Media Mol Imaging. 2018.
PMID: 29967572
Free PMC article.
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In Vivo Imaging of Local Inflammation: Monitoring LPS-Induced CD80/CD86 Upregulation by PET.
Taddio MF, Castro Jaramillo CA, Runge P, Blanc A, Keller C, Talip Z, Béhé M, van der Meulen NP, Halin C, Schibli R, Krämer SD.
Taddio MF, et al.
Mol Imaging Biol. 2021 Apr;23(2):196-207. doi: 10.1007/s11307-020-01543-3. Epub 2020 Sep 28.
Mol Imaging Biol. 2021.
PMID: 32989622
Free PMC article.
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