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Zhou Z, Zhou G, Zhou C, Fan Z, Cui R, Li Y, Li R, Gu Y, Li H, Ge Z, Cai X, Jiang B, Wang D, Zheng M, Xu T, Zhang S.
Zhou Z, et al. Among authors: cai x.
J Med Chem. 2023 Mar 23;66(6):4197-4214. doi: 10.1021/acs.jmedchem.3c00075. Epub 2023 Mar 10.
J Med Chem. 2023.
PMID: 36897932