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Powerful Potential of Polyfluoroalkyl-Containing 4-Arylhydrazinylidenepyrazol-3-ones for Pharmaceuticals.
Burgart YV, Elkina NA, Shchegolkov EV, Krasnykh OP, Makhaeva GF, Triandafilova GA, Solodnikov SY, Boltneva NP, Rudakova EV, Kovaleva NV, Serebryakova OG, Ulitko MV, Borisevich SS, Gerasimova NA, Evstigneeva NP, Kozlov SA, Korolkova YV, Minin AS, Belousova AV, Mozhaitsev ES, Klabukov AM, Saloutin VI. Burgart YV, et al. Among authors: kozlov sa. Molecules. 2022 Dec 21;28(1):59. doi: 10.3390/molecules28010059. Molecules. 2022. PMID: 36615256 Free PMC article.
Polypeptide modulators of TRPV1 produce analgesia without hyperthermia.
Andreev YA, Kozlov SA, Korolkova YV, Dyachenko IA, Bondarenko DA, Skobtsov DI, Murashev AN, Kotova PD, Rogachevskaja OA, Kabanova NV, Kolesnikov SS, Grishin EV. Andreev YA, et al. Among authors: kozlov sa. Mar Drugs. 2013 Dec 16;11(12):5100-15. doi: 10.3390/md11125100. Mar Drugs. 2013. PMID: 24351908 Free PMC article.
New Disulfide-Stabilized Fold Provides Sea Anemone Peptide to Exhibit Both Antimicrobial and TRPA1 Potentiating Properties.
Logashina YA, Solstad RG, Mineev KS, Korolkova YV, Mosharova IV, Dyachenko IA, Palikov VA, Palikova YA, Murashev AN, Arseniev AS, Kozlov SA, Stensvåg K, Haug T, Andreev YA. Logashina YA, et al. Among authors: kozlov sa. Toxins (Basel). 2017 Apr 29;9(5):154. doi: 10.3390/toxins9050154. Toxins (Basel). 2017. PMID: 28468269 Free PMC article.
TRPV1 activation power can switch an action mode for its polypeptide ligands.
Nikolaev MV, Dorofeeva NA, Komarova MS, Korolkova YV, Andreev YA, Mosharova IV, Grishin EV, Tikhonov DB, Kozlov SA. Nikolaev MV, et al. Among authors: kozlov sa. PLoS One. 2017 May 5;12(5):e0177077. doi: 10.1371/journal.pone.0177077. eCollection 2017. PLoS One. 2017. PMID: 28475608 Free PMC article.
5-Alkoxy-1-aryl-3-polyfluoroalkylpyrazoles with Antinociceptive Activity: Partial Agonists of TRPV1 Ion Channels.
Khudina OG, Burgart YV, Malkova NA, Shchegolkov EV, Krasnykh OP, Triandafilova GA, Malysheva KO, Solodnikov SY, Dubodel ES, Korolkova YV, Kozlov SA, Borisevich SS, Mozhaitsev ES, Saloutin VI. Khudina OG, et al. Among authors: kozlov sa. ChemMedChem. 2023 Jun 15;18(12):e202300063. doi: 10.1002/cmdc.202300063. Epub 2023 Apr 17. ChemMedChem. 2023. PMID: 37006199
154 results