Kapus GL - Search Results

1

Novel imidazo[1,5-a]quinoxaline derivatives: SAR, selectivity and modeling challenges en route to the identification of an α5-GABAA receptor NAM.

Károlyi BI, Potor A, Kapus GL, Fodor L, Bobok A, Krámos B, Magdó I, Bata I, Szabó G. Károlyi BI, et al. Among authors: kapus gl. Bioorg Med Chem Lett. 2023 Jan 15;80:129107. doi: 10.1016/j.bmcl.2022.129107. Epub 2022 Dec 19. Bioorg Med Chem Lett. 2023. PMID: 36549396

2

Multiparameter Optimization of Naphthyridine Derivatives as Selective α5-GABA_A Receptor Negative Allosteric Modulators.

Szabó G, Éliás O, Erdélyi P, Potor A, Túrós GI, Károlyi BI, Varró G, Vaskó ÁG, Bata I, Kapus GL, Dohányos Z, Bobok AÁ, Fodor L, Thán M, Vastag M, Komlódi Z, Soukupné Kedves RÉ, Makó É, Süveges B, Greiner I. Szabó G, et al. Among authors: kapus gl. J Med Chem. 2022 Jun 9;65(11):7876-7895. doi: 10.1021/acs.jmedchem.2c00414. Epub 2022 May 18. J Med Chem. 2022. PMID: 35584373

3

Identification of Triazolopyridines as Selective α5-GABA_A Receptor Negative Allosteric Modulators by a Hybridization Approach.

Szabó G, Károlyi BI, Vaskó ÁG, Potor A, Vukics K, Kapus GL, Fodor L, Bobok A, Vastag M, Bata I. Szabó G, et al. Among authors: kapus gl. ACS Chem Neurosci. 2023 Jan 4;14(1):148-158. doi: 10.1021/acschemneuro.2c00608. Epub 2022 Dec 16. ACS Chem Neurosci. 2023. PMID: 36524695

4

New non competitive AMPA antagonists.

Abrahám G, Sólyom S, Csuzdi E, Berzsenyi P, Ling I, Tarnawa I, Hámori T, Pallagi I, Horváth K, Andrási F, Kapus G, Hársing LG Jr, Király I, Patthy M, Horváth G. Abrahám G, et al. Bioorg Med Chem. 2000 Aug;8(8):2127-43. doi: 10.1016/s0968-0896(00)00133-4. Bioorg Med Chem. 2000. PMID: 11003158

5

Neuroprotective and anticonvulsant effects of EGIS-8332, a non-competitive AMPA receptor antagonist, in a range of animal models.

Gigler G, Móricz K, Agoston M, Simó A, Albert M, Benedek A, Kapus G, Kertész S, Vegh M, Barkóczy J, Markó B, Szabó G, Matucz E, Gacsályi I, Lévay G, Hársing LG Jr, Szénási G. Gigler G, et al. Br J Pharmacol. 2007 Sep;152(1):151-60. doi: 10.1038/sj.bjp.0707362. Epub 2007 Jul 2. Br J Pharmacol. 2007. PMID: 17603549 Free PMC article.

6

A novel GABA(A) alpha 5 receptor inhibitor with therapeutic potential.

Ling I, Mihalik B, Etherington LA, Kapus G, Pálvölgyi A, Gigler G, Kertész S, Gaál A, Pallagi K, Kiricsi P, Szabó É, Szénási G, Papp L, Hársing LG, Lévay G, Spedding M, Lambert JJ, Belelli D, Barkóczy J, Volk B, Simig G, Gacsályi I, Antoni FA. Ling I, et al. Eur J Pharmacol. 2015 Oct 5;764:497-507. doi: 10.1016/j.ejphar.2015.07.005. Epub 2015 Jul 11. Eur J Pharmacol. 2015. PMID: 26169564

7

Differential modulation of the GYKI 53784-induced inhibition of AMPA currents by various AMPA-positive modulators in cerebellar Purkinje cells.

Kapus G, Bódi I, Pataki A, Gueritaud J, Székely JI, Tarnawa I. Kapus G, et al. Eur J Pharmacol. 2000 May 26;397(1):43-7. doi: 10.1016/s0014-2999(00)00302-2. Eur J Pharmacol. 2000. PMID: 10844097

8

Converging Evidence on D-Amino Acid Oxidase-Dependent Enhancement of Hippocampal Firing Activity and Passive Avoidance Learning in Rats.

Nagy LV, Bali ZK, Kapus G, Pelsőczi P, Farkas B, Lendvai B, Lévay G, Hernádi I. Nagy LV, et al. Int J Neuropsychopharmacol. 2021 May 18;24(5):434-445. doi: 10.1093/ijnp/pyaa095. Int J Neuropsychopharmacol. 2021. PMID: 33305805 Free PMC article.

9

Antagonism of AMPA receptors produces anxiolytic-like behavior in rodents: effects of GYKI 52466 and its novel analogues.

Kapus GL, Gacsályi I, Vegh M, Kompagne H, Hegedus E, Leveleki C, Hársing LG, Barkóczy J, Bilkei-Gorzó A, Lévay G. Kapus GL, et al. Psychopharmacology (Berl). 2008 Jun;198(2):231-41. doi: 10.1007/s00213-008-1121-z. Epub 2008 Mar 25. Psychopharmacology (Berl). 2008. PMID: 18363046

10

2,3-benzodiazepine-type AMPA receptor antagonists and their neuroprotective effects.

Szénási G, Vegh M, Szabo G, Kertesz S, Kapus G, Albert M, Greff Z, Ling I, Barkoczy J, Simig G, Spedding M, Harsing LG Jr. Szénási G, et al. Neurochem Int. 2008 Jan;52(1-2):166-83. doi: 10.1016/j.neuint.2007.07.002. Epub 2007 Jul 10. Neurochem Int. 2008. PMID: 17707550 Review.

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