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Discovery of JNJ-64264681: A Potent and Selective Covalent Inhibitor of Bruton's Tyrosine Kinase.
J Med Chem. 2022 Nov 10;65(21):14326-14336. doi: 10.1021/acs.jmedchem.2c01026. Epub 2022 Oct 31.
J Med Chem. 2022.
PMID: 36314537
Citrullination/Methylation Crosstalk on Histone H3 Regulates ER-Target Gene Transcription.
Clancy KW, Russell AM, Subramanian V, Nguyen H, Qian Y, Campbell RM, Thompson PR.
Clancy KW, et al.
ACS Chem Biol. 2017 Jun 16;12(6):1691-1702. doi: 10.1021/acschembio.7b00241. Epub 2017 May 9.
ACS Chem Biol. 2017.
PMID: 28485572
Free PMC article.
Item in Clipboard
Detection and identification of protein citrullination in complex biological systems.
Clancy KW, Weerapana E, Thompson PR.
Clancy KW, et al.
Curr Opin Chem Biol. 2016 Feb;30:1-6. doi: 10.1016/j.cbpa.2015.10.014. Epub 2015 Oct 27.
Curr Opin Chem Biol. 2016.
PMID: 26517730
Free PMC article.
Review.
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Chemical Proteomic Platform To Identify Citrullinated Proteins.
Lewallen DM, Bicker KL, Subramanian V, Clancy KW, Slade DJ, Martell J, Dreyton CJ, Sokolove J, Weerapana E, Thompson PR.
Lewallen DM, et al. Among authors: clancy kw.
ACS Chem Biol. 2015 Nov 20;10(11):2520-8. doi: 10.1021/acschembio.5b00438. Epub 2015 Sep 23.
ACS Chem Biol. 2015.
PMID: 26360112
Free PMC article.
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Chemical biology of protein arginine modifications in epigenetic regulation.
Fuhrmann J, Clancy KW, Thompson PR.
Fuhrmann J, et al. Among authors: clancy kw.
Chem Rev. 2015 Jun 10;115(11):5413-61. doi: 10.1021/acs.chemrev.5b00003. Epub 2015 May 13.
Chem Rev. 2015.
PMID: 25970731
Free PMC article.
Review.
No abstract available.
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Autocatalytic intramolecular isopeptide bond formation in gram-positive bacterial pili: a QM/MM simulation.
Hu X, Hu H, Melvin JA, Clancy KW, McCafferty DG, Yang W.
Hu X, et al. Among authors: clancy kw.
J Am Chem Soc. 2011 Jan 26;133(3):478-85. doi: 10.1021/ja107513t. Epub 2010 Dec 13.
J Am Chem Soc. 2011.
PMID: 21142157
Free PMC article.
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Sortase transpeptidases: insights into mechanism, substrate specificity, and inhibition.
Clancy KW, Melvin JA, McCafferty DG.
Clancy KW, et al.
Biopolymers. 2010;94(4):385-96. doi: 10.1002/bip.21472.
Biopolymers. 2010.
PMID: 20593474
Free PMC article.
Review.
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NMDA receptor-nitric oxide transmission mediates neuronal iron homeostasis via the GTPase Dexras1.
Cheah JH, Kim SF, Hester LD, Clancy KW, Patterson SE 3rd, Papadopoulos V, Snyder SH.
Cheah JH, et al. Among authors: clancy kw.
Neuron. 2006 Aug 17;51(4):431-40. doi: 10.1016/j.neuron.2006.07.011.
Neuron. 2006.
PMID: 16908409
Free PMC article.
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