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Highly Potent and Oral Macrocyclic Peptides as a HIV-1 Protease Inhibitor: mRNA Display-Derived Hit-to-Lead Optimization.
ACS Med Chem Lett. 2022 Sep 1;13(10):1634-1641. doi: 10.1021/acsmedchemlett.2c00310. eCollection 2022 Oct 13.
ACS Med Chem Lett. 2022.
PMID: 36262395
Free PMC article.
Stalobacin: Discovery of Novel Lipopeptide Antibiotics with Potent Antibacterial Activity against Multidrug-Resistant Bacteria.
Matsui K, Kan Y, Kikuchi J, Matsushima K, Takemura M, Maki H, Kozono I, Ueda T, Minagawa K.
Matsui K, et al. Among authors: kozono i.
J Med Chem. 2020 Jun 11;63(11):6090-6095. doi: 10.1021/acs.jmedchem.0c00295. Epub 2020 May 19.
J Med Chem. 2020.
PMID: 32378891
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Peptide-to-Small Molecule: Discovery of Non-Covalent, Active-Site Inhibitors of β-Herpesvirus Proteases.
Yoshida S, Sako Y, Nikaido E, Ueda T, Kozono I, Ichihashi Y, Nakahashi A, Onishi M, Yamatsu Y, Kato T, Nishikawa J, Tachibana Y.
Yoshida S, et al. Among authors: kozono i.
ACS Med Chem Lett. 2023 Oct 27;14(11):1558-1566. doi: 10.1021/acsmedchemlett.3c00359. eCollection 2023 Nov 9.
ACS Med Chem Lett. 2023.
PMID: 37974946
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Engineering of the cytochrome P450 monooxygenase system for benzyl maltol hydroxylation.
Kozono I, Mihara K, Minagawa K, Hibi M, Ogawa J.
Kozono I, et al.
Appl Microbiol Biotechnol. 2017 Sep;101(17):6651-6658. doi: 10.1007/s00253-017-8414-2. Epub 2017 Jul 20.
Appl Microbiol Biotechnol. 2017.
PMID: 28730410
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Purification and characterization of molybdenum-containing aldehyde dehydrogenase that oxidizes benzyl maltol derivative from Pseudomonas nitroreducens SB32154.
Kozono I, Hibi M, Takeuchi M, Ogawa J.
Kozono I, et al.
Biosci Biotechnol Biochem. 2020 Nov;84(11):2390-2400. doi: 10.1080/09168451.2020.1799749. Epub 2020 Jul 30.
Biosci Biotechnol Biochem. 2020.
PMID: 32729393
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Characterization of xanthine oxidase from Cellulosimicrobium funkei possessing hypoxanthine-metabolizing activity.
Kozono I, Takeuchi M, Kozono S, Satomura A, Aoki W, Hibi M, Ogawa J.
Kozono I, et al.
J Appl Microbiol. 2021 Jun;130(6):2132-2140. doi: 10.1111/jam.14891. Epub 2020 Nov 22.
J Appl Microbiol. 2021.
PMID: 33090589
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