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Characterization of Dual-Acting A3 Adenosine Receptor Positive Allosteric Modulators That Preferentially Enhance Adenosine-Induced Gαi3 and GαoA Isoprotein Activation.
ACS Pharmacol Transl Sci. 2022 Jul 15;5(8):625-641. doi: 10.1021/acsptsci.2c00076. eCollection 2022 Aug 12.
ACS Pharmacol Transl Sci. 2022.
PMID: 35983277
Free PMC article.
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Structure-Activity Studies of 1H-Imidazo[4,5-c]quinolin-4-amine Derivatives as A3 Adenosine Receptor Positive Allosteric Modulators.
Fallot LB, Suresh RR, Fisher CL, Salmaso V, O'Connor RD, Kaufman N, Gao ZG, Auchampach JA, Jacobson KA.
Fallot LB, et al.
J Med Chem. 2022 Nov 24;65(22):15238-15262. doi: 10.1021/acs.jmedchem.2c01170. Epub 2022 Nov 11.
J Med Chem. 2022.
PMID: 36367749
Free PMC article.
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