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A Novel Triple-Action Inhibitor Targeting B-Cell Receptor Signaling and BRD4 Demonstrates Preclinical Activity in Chronic Lymphocytic Leukemia.
Int J Mol Sci. 2022 Jun 16;23(12):6712. doi: 10.3390/ijms23126712.
Int J Mol Sci. 2022.
PMID: 35743155
Free PMC article.
Preclinical activity of a novel multi-axis inhibitor in aggressive and indolent B-cell malignancies.
Smith AL, Pal D, Martinez-Rico R, Eiken AP, Durden DL, Kutateladze TG, El-Gamal D.
Smith AL, et al. Among authors: eiken ap.
Leuk Lymphoma. 2023 Dec;64(14):2333-2337. doi: 10.1080/10428194.2023.2256914. Epub 2023 Sep 14.
Leuk Lymphoma. 2023.
PMID: 37706519
No abstract available.
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BET inhibition reforms the immune microenvironment and alleviates T cell dysfunction in chronic lymphocytic leukemia.
Smith AL, Skupa SA, Eiken AP, Reznicek TE, Schmitz E, Williams N, Moore DY, D'Angelo CR, Kallam A, Lunning MA, Bociek RG, Vose JM, Mohamed E, Mahr AR, Denton PW, Powell B, Bollag G, Rowley MJ, El-Gamal D.
Smith AL, et al. Among authors: eiken ap.
JCI Insight. 2024 May 22;9(10):e177054. doi: 10.1172/jci.insight.177054.
JCI Insight. 2024.
PMID: 38775157
Free PMC article.
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Novel Spirocyclic Dimer, SpiD3, Targets Chronic Lymphocytic Leukemia Survival Pathways with Potent Preclinical Effects.
Eiken AP, Smith AL, Skupa SA, Schmitz E, Rana S, Singh S, Kumar S, Mallareddy JR, de Cubas AA, Krishna A, Kalluchi A, Rowley MJ, D'Angelo CR, Lunning MA, Bociek RG, Vose JM, Natarajan A, El-Gamal D.
Eiken AP, et al.
Cancer Res Commun. 2024 May 22;4(5):1328-1343. doi: 10.1158/2767-9764.CRC-24-0071.
Cancer Res Commun. 2024.
PMID: 38687198
Free PMC article.
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Editorial for the IJMS Special Issue on Molecular Pathogenesis and Molecular Therapy of Lymphoid Malignancies.
Eiken AP, El-Gamal D.
Eiken AP, et al.
Int J Mol Sci. 2023 Dec 31;25(1):557. doi: 10.3390/ijms25010557.
Int J Mol Sci. 2023.
PMID: 38203728
Free PMC article.
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