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Bioactivity of Novel Pyrazole-Thiazolines Scaffolds against Trypanosoma cruzi: Computational Approaches and 3D Spheroid Model on Drug Discovery for Chagas Disease.
Pharmaceutics. 2022 May 5;14(5):995. doi: 10.3390/pharmaceutics14050995.
Pharmaceutics. 2022.
PMID: 35631581
Free PMC article.
Structural Optimization and Biological Activity of Pyrazole Derivatives: Virtual Computational Analysis, Recovery Assay and 3D Culture Model as Potential Predictive Tools of Effectiveness against Trypanosoma cruzi.
Orlando LMR, Lechuga GC, da Silva Lara L, Ferreira BS, Pereira CN, Silva RC, Dos Santos MS, Pereira MCS.
Orlando LMR, et al.
Molecules. 2021 Nov 8;26(21):6742. doi: 10.3390/molecules26216742.
Molecules. 2021.
PMID: 34771151
Free PMC article.
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Antitrypanosomal Activity of 1,2,3-Triazole-Based Hybrids Evaluated Using In Vitro Preclinical Translational Models.
Orlando LMR, Lara LDS, Lechuga GC, Rodrigues GC, Pandoli OG, de Sá DS, Pereira MCS.
Orlando LMR, et al.
Biology (Basel). 2023 Sep 8;12(9):1222. doi: 10.3390/biology12091222.
Biology (Basel). 2023.
PMID: 37759621
Free PMC article.
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