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Thietanes and Derivatives thereof in Medicinal Chemistry.
Francisco KR, Ballatore C. Francisco KR, et al. Among authors: ballatore c. Curr Top Med Chem. 2022;22(15):1219-1234. doi: 10.2174/1568026622666220511154228. Curr Top Med Chem. 2022. PMID: 35546768 Review.
Structure Property Relationships of Carboxylic Acid Isosteres.
Lassalas P, Gay B, Lasfargeas C, James MJ, Tran V, Vijayendran KG, Brunden KR, Kozlowski MC, Thomas CJ, Smith AB 3rd, Huryn DM, Ballatore C. Lassalas P, et al. Among authors: ballatore c. J Med Chem. 2016 Apr 14;59(7):3183-203. doi: 10.1021/acs.jmedchem.5b01963. Epub 2016 Mar 30. J Med Chem. 2016. PMID: 26967507 Free PMC article.
Evaluation of Oxetan-3-ol, Thietan-3-ol, and Derivatives Thereof as Bioisosteres of the Carboxylic Acid Functional Group.
Lassalas P, Oukoloff K, Makani V, James M, Tran V, Yao Y, Huang L, Vijayendran K, Monti L, Trojanowski JQ, Lee VM, Kozlowski MC, Smith AB 3rd, Brunden KR, Ballatore C. Lassalas P, et al. Among authors: ballatore c. ACS Med Chem Lett. 2017 Jul 5;8(8):864-868. doi: 10.1021/acsmedchemlett.7b00212. eCollection 2017 Aug 10. ACS Med Chem Lett. 2017. PMID: 28835803 Free PMC article.
Design, synthesis and evaluation of photoactivatable derivatives of microtubule (MT)-active [1,2,4]triazolo[1,5-a]pyrimidines.
Oukoloff K, Kovalevich J, Cornec AS, Yao Y, Owyang ZA, James M, Trojanowski JQ, Lee VM, Smith AB 3rd, Brunden KR, Ballatore C. Oukoloff K, et al. Among authors: ballatore c. Bioorg Med Chem Lett. 2018 Jul 1;28(12):2180-2183. doi: 10.1016/j.bmcl.2018.05.010. Epub 2018 May 5. Bioorg Med Chem Lett. 2018. PMID: 29764743 Free PMC article.
1,2,4-Triazolo[1,5-a]pyrimidines in drug design.
Oukoloff K, Lucero B, Francisco KR, Brunden KR, Ballatore C. Oukoloff K, et al. Among authors: ballatore c. Eur J Med Chem. 2019 Mar 1;165:332-346. doi: 10.1016/j.ejmech.2019.01.027. Epub 2019 Jan 14. Eur J Med Chem. 2019. PMID: 30703745 Free PMC article. Review.
Evaluation of the Structure-Activity Relationship of Microtubule-Targeting 1,2,4-Triazolo[1,5-a]pyrimidines Identifies New Candidates for Neurodegenerative Tauopathies.
Oukoloff K, Nzou G, Varricchio C, Lucero B, Alle T, Kovalevich J, Monti L, Cornec AS, Yao Y, James MJ, Trojanowski JQ, Lee VM, Smith AB 3rd, Brancale A, Brunden KR, Ballatore C. Oukoloff K, et al. Among authors: ballatore c. J Med Chem. 2021 Jan 28;64(2):1073-1102. doi: 10.1021/acs.jmedchem.0c01605. Epub 2021 Jan 7. J Med Chem. 2021. PMID: 33411523 Free PMC article.
Inhibition of the HEG1-KRIT1 interaction increases KLF4 and KLF2 expression in endothelial cells.
Lopez-Ramirez MA, McCurdy S, Li W, Haynes MK, Hale P, Francisco K, Oukoloff K, Bautista M, Choi CHJ, Sun H, Gongol B, Shyy JY, Ballatore C, Sklar LA, Gingras AR. Lopez-Ramirez MA, et al. Among authors: ballatore c. FASEB Bioadv. 2021 Feb 18;3(5):334-355. doi: 10.1096/fba.2020-00141. eCollection 2021 May. FASEB Bioadv. 2021. PMID: 33977234 Free PMC article.
Evaluation of log P, pKa, and log D predictions from the SAMPL7 blind challenge.
Bergazin TD, Tielker N, Zhang Y, Mao J, Gunner MR, Francisco K, Ballatore C, Kast SM, Mobley DL. Bergazin TD, et al. Among authors: ballatore c. J Comput Aided Mol Des. 2021 Jul;35(7):771-802. doi: 10.1007/s10822-021-00397-3. Epub 2021 Jun 24. J Comput Aided Mol Des. 2021. PMID: 34169394 Free PMC article.
79 results