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Dihydropyridine Lactam Analogs Targeting BET Bromodomains.
Jiang J, Sigua LH, Chan A, Kalra P, Pomerantz WCK, Schönbrunn E, Qi J, Georg GI. Jiang J, et al. Among authors: pomerantz wck. ChemMedChem. 2022 Jan 5;17(1):e202100407. doi: 10.1002/cmdc.202100407. Epub 2021 Dec 21. ChemMedChem. 2022. PMID: 34932262 Free PMC article.
Genetically encoded discovery of perfluoroaryl macrocycles that bind to albumin and exhibit extended circulation in vivo.
Wong JYK, Ekanayake AI, Kharchenko S, Kirberger SE, Qiu R, Kelich P, Sarkar S, Li J, Fernandez KX, Alvizo-Paez ER, Miao J, Kalhor-Monfared S, John JD, Kang H, Choi H, Nuss JM, Vederas JC, Lin YS, Macauley MS, Vukovic L, Pomerantz WCK, Derda R. Wong JYK, et al. Among authors: pomerantz wck. Nat Commun. 2023 Sep 13;14(1):5654. doi: 10.1038/s41467-023-41427-y. Nat Commun. 2023. PMID: 37704629 Free PMC article.
BET Bromodomain Inhibitors with One-Step Synthesis Discovered from Virtual Screen.
Ayoub AM, Hawk LML, Herzig RJ, Jiang J, Wisniewski AJ, Gee CT, Zhao P, Zhu JY, Berndt N, Offei-Addo NK, Scott TG, Qi J, Bradner JE, Ward TR, Schönbrunn E, Georg GI, Pomerantz WCK. Ayoub AM, et al. Among authors: pomerantz wck. J Med Chem. 2017 Jun 22;60(12):4805-4817. doi: 10.1021/acs.jmedchem.6b01336. Epub 2017 Jun 7. J Med Chem. 2017. PMID: 28535045 Free PMC article.
Correction to BET Bromodomain Inhibitors with One-Step Synthesis Discovered from Virtual Screen.
Ayoub AM, Hawk LML, Herzig RJ, Jiang J, Wisniewski AJ, Gee CT, Zhao P, Zhu JY, Berndt N, Offei-Addo NK, Scott TG, Qi J, Bradner JE, Ward TR, Schönbrunn E, Georg GI, Pomerantz WCK. Ayoub AM, et al. Among authors: pomerantz wck. J Med Chem. 2017 Jul 27;60(14):6458. doi: 10.1021/acs.jmedchem.7b00943. Epub 2017 Jul 11. J Med Chem. 2017. PMID: 28696689 No abstract available.
Molecular Basis for the N-Terminal Bromodomain-and-Extra-Terminal-Family Selectivity of a Dual Kinase-Bromodomain Inhibitor.
Divakaran A, Talluri SK, Ayoub AM, Mishra NK, Cui H, Widen JC, Berndt N, Zhu JY, Carlson AS, Topczewski JJ, Schonbrunn EK, Harki DA, Pomerantz WCK. Divakaran A, et al. Among authors: pomerantz wck. J Med Chem. 2018 Oct 25;61(20):9316-9334. doi: 10.1021/acs.jmedchem.8b01248. Epub 2018 Oct 16. J Med Chem. 2018. PMID: 30253095 Free PMC article.
SAR by (Protein-Observed) 19F NMR.
Divakaran A, Kirberger SE, Pomerantz WCK. Divakaran A, et al. Among authors: pomerantz wck. Acc Chem Res. 2019 Dec 17;52(12):3407-3418. doi: 10.1021/acs.accounts.9b00377. Epub 2019 Nov 13. Acc Chem Res. 2019. PMID: 31718149 Free PMC article. Review.
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