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Synthesis, Characterization, and Preclinical Evaluation of a Small-Molecule Prostate-Specific Membrane Antigen-Targeted Monomethyl Auristatin E Conjugate.
J Med Chem. 2021 Dec 9;64(23):17123-17145. doi: 10.1021/acs.jmedchem.1c01157. Epub 2021 Nov 19.
J Med Chem. 2021.
PMID: 34797052
PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation.
Machulkin AE, Uspenskaya AA, Zyk NY, Nimenko EA, Ber AP, Petrov SA, Shafikov RR, Skvortsov DA, Smirnova GB, Borisova YA, Pokrovsky VS, Kolmogorov VS, Vaneev AN, Ivanenkov YA, Khudyakov AD, Kovalev SV, Erofeev AS, Gorelkin PV, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG.
Machulkin AE, et al. Among authors: khudyakov ad.
Eur J Med Chem. 2022 Jan 5;227:113936. doi: 10.1016/j.ejmech.2021.113936. Epub 2021 Oct 23.
Eur J Med Chem. 2022.
PMID: 34717125
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Design and synthesis of atorvastatin derivatives with enhanced water solubility, hepatoselectivity and stability.
Maklakova SY, Lopukhov AV, Khudyakov AD, Kovalev SV, Mazhuga MP, Chepikova OE, Zamyatnin AA Jr, Majouga AG, Klyachko NL, Beloglazkina EK.
Maklakova SY, et al. Among authors: khudyakov ad.
RSC Med Chem. 2022 Oct 11;14(1):56-64. doi: 10.1039/d2md00119e. eCollection 2023 Jan 25.
RSC Med Chem. 2022.
PMID: 36760736
Free PMC article.
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