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Novel imidazo[2,1-b]thiazole-based anticancer agents as potential focal adhesion kinase inhibitors: Synthesis, in silico and in vitro evaluation.
Chem Biol Drug Des. 2021 Aug;98(2):270-282. doi: 10.1111/cbdd.13896. Epub 2021 Jun 12.
Chem Biol Drug Des. 2021.
PMID: 34021971
Design and synthesis of novel Imidazo[2,1-b]thiazole derivatives as potent antiviral and antimycobacterial agents.
Gürsoy E, Dincel ED, Naesens L, Ulusoy Güzeldemirci N.
Gürsoy E, et al. Among authors: ulusoy guzeldemirci n.
Bioorg Chem. 2020 Jan;95:103496. doi: 10.1016/j.bioorg.2019.103496. Epub 2019 Dec 6.
Bioorg Chem. 2020.
PMID: 31862455
Free PMC article.
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Antioxidant activity of novel imidazo[2,1-b]thiazole derivatives: Design, synthesis, biological evaluation, molecular docking study and in silico ADME prediction.
Dincel ED, Gürsoy E, Yilmaz-Ozden T, Ulusoy-Güzeldemirci N.
Dincel ED, et al. Among authors: ulusoy guzeldemirci n.
Bioorg Chem. 2020 Oct;103:104220. doi: 10.1016/j.bioorg.2020.104220. Epub 2020 Aug 26.
Bioorg Chem. 2020.
PMID: 32896742
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Synthesis and Aldose Reductase Inhibitory Effect of Some New Hydrazinecarbothioamides and 4-Thiazolidinones Bearing an Imidazo[2,1-b]Thiazole Moiety.
Ulusoy Güzeldemirci N, Cimok S, Daş-Evcimen N, Sarikaya M.
Ulusoy Güzeldemirci N, et al.
Turk J Pharm Sci. 2019 Mar;16(1):1-7. doi: 10.4274/tjps.05900. Epub 2018 Dec 31.
Turk J Pharm Sci. 2019.
PMID: 32454687
Free PMC article.
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Antibacterial, Antitubercular and Antiviral Activity Evaluations of Some Arylidenehydrazide Derivatives Bearing Imidazo[2,1-b]thiazole Moiety.
Ulusoy Güzeldemirci N, Karaman B, Küçükbasmaci Ö.
Ulusoy Güzeldemirci N, et al.
Turk J Pharm Sci. 2017 Aug;14(2):157-163. doi: 10.4274/tjps.25743. Epub 2017 Aug 15.
Turk J Pharm Sci. 2017.
PMID: 32454607
Free PMC article.
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Synthesis and antiviral properties of novel indole-based thiosemicarbazides and 4-thiazolidinones.
Cihan-Üstündağ G, Gürsoy E, Naesens L, Ulusoy-Güzeldemirci N, Çapan G.
Cihan-Üstündağ G, et al. Among authors: ulusoy guzeldemirci n.
Bioorg Med Chem. 2016 Jan 15;24(2):240-6. doi: 10.1016/j.bmc.2015.12.008. Epub 2015 Dec 8.
Bioorg Med Chem. 2016.
PMID: 26707844
Free PMC article.
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Design, synthesis, and evaluation of novel bistrifluoromethyl-based hydrazones as dual inhibitors of acetylcholinesterase and carbonic anhydrase enzymes for Alzheimer's disease.
Dincel ED, Başoğlu-Ünal F, Kuran ED, Kayra T, Aydın N, Kanber E, Gülçin İ, Ulusoy-Güzeldemirci N.
Dincel ED, et al. Among authors: ulusoy guzeldemirci n.
Chem Biol Drug Des. 2024 Feb;103(2):e14482. doi: 10.1111/cbdd.14482.
Chem Biol Drug Des. 2024.
PMID: 38378259
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