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Macrocyclic Peptides that Selectively Inhibit the Mycobacterium tuberculosis Proteasome.
J Med Chem. 2021 May 13;64(9):6262-6272. doi: 10.1021/acs.jmedchem.1c00296. Epub 2021 May 5.
J Med Chem. 2021.
PMID: 33949190
Free PMC article.
Development of a Highly Selective Plasmodium falciparum Proteasome Inhibitor with Anti-malaria Activity in Humanized Mice.
Zhan W, Zhang H, Ginn J, Leung A, Liu YJ, Michino M, Toita A, Okamoto R, Wong TT, Imaeda T, Hara R, Yukawa T, Chelebieva S, Tumwebaze PK, Lafuente-Monasterio MJ, Martinez-Martinez MS, Vendome J, Beuming T, Sato K, Aso K, Rosenthal PJ, Cooper RA, Meinke PT, Nathan CF, Kirkman LA, Lin G.
Zhan W, et al. Among authors: toita a.
Angew Chem Int Ed Engl. 2021 Apr 19;60(17):9279-9283. doi: 10.1002/anie.202015845. Epub 2021 Mar 11.
Angew Chem Int Ed Engl. 2021.
PMID: 33433953
Free PMC article.
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Design, Synthesis, and Optimization of Macrocyclic Peptides as Species-Selective Antimalaria Proteasome Inhibitors.
Zhang H, Ginn J, Zhan W, Liu YJ, Leung A, Toita A, Okamoto R, Wong TT, Imaeda T, Hara R, Yukawa T, Michino M, Vendome J, Beuming T, Sato K, Aso K, Meinke PT, Nathan CF, Kirkman LA, Lin G.
Zhang H, et al. Among authors: toita a.
J Med Chem. 2022 Jul 14;65(13):9350-9375. doi: 10.1021/acs.jmedchem.2c00611. Epub 2022 Jun 21.
J Med Chem. 2022.
PMID: 35727231
Free PMC article.
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Discovery of 3-Benzyl-1-( trans-4-((5-cyanopyridin-2-yl)amino)cyclohexyl)-1-arylurea Derivatives as Novel and Selective Cyclin-Dependent Kinase 12 (CDK12) Inhibitors.
Ito M, Tanaka T, Toita A, Uchiyama N, Kokubo H, Morishita N, Klein MG, Zou H, Murakami M, Kondo M, Sameshima T, Araki S, Endo S, Kawamoto T, Morin GB, Aparicio SA, Nakanishi A, Maezaki H, Imaeda Y.
Ito M, et al. Among authors: toita a.
J Med Chem. 2018 Sep 13;61(17):7710-7728. doi: 10.1021/acs.jmedchem.8b00683. Epub 2018 Aug 20.
J Med Chem. 2018.
PMID: 30067358
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Total syntheses of (+)-polygalolide a and (+)-polygalolide b: elucidation of the absolute stereochemistry and biogenetic implications.
Sugano Y, Kikuchi F, Toita A, Nakamura S, Hashimoto S.
Sugano Y, et al. Among authors: toita a.
Chemistry. 2012 Jul 27;18(31):9682-90. doi: 10.1002/chem.201200542. Epub 2012 Jul 3.
Chemistry. 2012.
PMID: 22760948
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Novel quinazolin-4(3H)-one based Cyclin K degraders regulate alternative polyadenylation activity.
Sano O, Ito M, Saito M, Toita A, Tanaka T, Maezaki H, Araki S, Iwata H.
Sano O, et al. Among authors: toita a.
Biochem Biophys Res Commun. 2023 Oct 8;676:6-12. doi: 10.1016/j.bbrc.2023.07.028. Epub 2023 Jul 17.
Biochem Biophys Res Commun. 2023.
PMID: 37480690
Free article.
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Structure-Activity Relationship Studies of Antimalarial Plasmodium Proteasome Inhibitors─Part II.
Zhang H, Ginn J, Zhan W, Leung A, Liu YJ, Toita A, Okamoto R, Wong TT, Imaeda T, Hara R, Michino M, Yukawa T, Chelebieva S, Tumwebaze PK, Vendome J, Beuming T, Sato K, Aso K, Rosenthal PJ, Cooper RA, Liverton N, Foley M, Meinke PT, Nathan CF, Kirkman LA, Lin G.
Zhang H, et al. Among authors: toita a.
J Med Chem. 2023 Jan 26;66(2):1484-1508. doi: 10.1021/acs.jmedchem.2c01651. Epub 2023 Jan 11.
J Med Chem. 2023.
PMID: 36630286
Free PMC article.
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