Kellam B - Search Results

1

Identification of a novel toxicophore in anti-cancer chemotherapeutics that targets mitochondrial respiratory complex I.

Stephenson ZA, Harvey RF, Pryde KR, Mistry S, Hardy RE, Serreli R, Chung I, Allen TE, Stoneley M, MacFarlane M, Fischer PM, Hirst J, Kellam B, Willis AE. Stephenson ZA, et al. Among authors: kellam b. Elife. 2020 May 20;9:e55845. doi: 10.7554/eLife.55845. Elife. 2020. PMID: 32432547 Free PMC article.

2

Immunosuppressive but non-LasR-inducing analogues of the Pseudomonas aeruginosa quorum-sensing molecule N-(3-oxododecanoyl)-l-homoserine lactone.

Jadhav GP, Chhabra SR, Telford G, Hooi DS, Righetti K, Williams P, Kellam B, Pritchard DI, Fischer PM. Jadhav GP, et al. Among authors: kellam b. J Med Chem. 2011 May 12;54(9):3348-59. doi: 10.1021/jm2001019. Epub 2011 Apr 13. J Med Chem. 2011. PMID: 21488685

3

Synthesis and in vitro and in vivo characterization of highly β1-selective β-adrenoceptor partial agonists.

Mistry SN, Baker JG, Fischer PM, Hill SJ, Gardiner SM, Kellam B. Mistry SN, et al. Among authors: kellam b. J Med Chem. 2013 May 23;56(10):3852-65. doi: 10.1021/jm400348g. Epub 2013 May 10. J Med Chem. 2013. PMID: 23614528 Free PMC article.

4

5-Deazaflavin derivatives as inhibitors of p53 ubiquitination by HDM2.

Dickens MP, Roxburgh P, Hock A, Mezna M, Kellam B, Vousden KH, Fischer PM. Dickens MP, et al. Among authors: kellam b. Bioorg Med Chem. 2013 Nov 15;21(22):6868-77. doi: 10.1016/j.bmc.2013.09.038. Epub 2013 Sep 25. Bioorg Med Chem. 2013. PMID: 24113239 Free PMC article.

5

GPCRs through the keyhole: the role of protein flexibility in ligand binding to β-adrenoceptors.

Emtage AL, Mistry SN, Fischer PM, Kellam B, Laughton CA. Emtage AL, et al. Among authors: kellam b. J Biomol Struct Dyn. 2017 Sep;35(12):2604-2619. doi: 10.1080/07391102.2016.1226197. Epub 2016 Sep 1. J Biomol Struct Dyn. 2017. PMID: 27532213

6

Novel selective β₁-adrenoceptor antagonists for concomitant cardiovascular and respiratory disease.

Baker JG, Gardiner SM, Woolard J, Fromont C, Jadhav GP, Mistry SN, Thompson KSJ, Kellam B, Hill SJ, Fischer PM. Baker JG, et al. Among authors: kellam b. FASEB J. 2017 Jul;31(7):3150-3166. doi: 10.1096/fj.201601305R. Epub 2017 Apr 11. FASEB J. 2017. PMID: 28400472 Free PMC article.

., Fromont, C., Jadhav, G. P., Mistry, S. N., Thompson, K. S. J., Kellam, B., Hill, S. J., Fischer, P. M. Novel selective beta(1)-adrenoceptor antagonists for concomitant cardiovascular and respiratory disease....

., Fromont, C., Jadhav, G. P., Mistry, S. N., Thompson, K. S. J., Kellam, B., Hill, S. J., Fischer, P. M. Novel selective beta …

7

Visualizing Ligand Binding to a GPCR In Vivo Using NanoBRET.

Alcobia DC, Ziegler AI, Kondrashov A, Comeo E, Mistry S, Kellam B, Chang A, Woolard J, Hill SJ, Sloan EK. Alcobia DC, et al. Among authors: kellam b. iScience. 2018 Aug 31;6:280-288. doi: 10.1016/j.isci.2018.08.006. Epub 2018 Aug 11. iScience. 2018. PMID: 30240618 Free PMC article.

8

Using Esterase Selectivity to Determine the In Vivo Duration of Systemic Availability and Abolish Systemic Side Effects of Topical β-Blockers.

Baker JG, Fromont C, Bruder M, Thompson KSJ, Kellam B, Hill SJ, Gardiner SM, Fischer PM. Baker JG, et al. Among authors: kellam b. ACS Pharmacol Transl Sci. 2020 Jul 1;3(4):737-748. doi: 10.1021/acsptsci.0c00051. eCollection 2020 Aug 14. ACS Pharmacol Transl Sci. 2020. PMID: 32832874 Free PMC article.

9

Subtype selective fluorescent ligands based on ICI 118,551 to study the human β2-adrenoceptor in CRISPR/Cas9 genome-edited HEK293T cells at low expression levels.

Goulding J, Mistry SJ, Soave M, Woolard J, Briddon SJ, White CW, Kellam B, Hill SJ. Goulding J, et al. Among authors: kellam b. Pharmacol Res Perspect. 2021 May;9(3):e00779. doi: 10.1002/prp2.779. Pharmacol Res Perspect. 2021. PMID: 34003582 Free PMC article.

10

Optimization of Peptide Linker-Based Fluorescent Ligands for the Histamine H₁ Receptor.

Kok ZY, Stoddart LA, Mistry SJ, Mocking TAM, Vischer HF, Leurs R, Hill SJ, Mistry SN, Kellam B. Kok ZY, et al. Among authors: kellam b. J Med Chem. 2022 Jun 23;65(12):8258-8288. doi: 10.1021/acs.jmedchem.2c00125. Epub 2022 Jun 3. J Med Chem. 2022. PMID: 35734860 Free PMC article.

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