Bretner M - Search Results

1

Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α' Structures.

Lindenblatt D, Nickelsen A, Applegate VM, Hochscherf J, Witulski B, Bouaziz Z, Marminon C, Bretner M, Le Borgne M, Jose J, Niefind K. Lindenblatt D, et al. Among authors: bretner m. ACS Omega. 2019 Mar 19;4(3):5471-5478. doi: 10.1021/acsomega.8b03415. eCollection 2019 Mar 31. ACS Omega. 2019. PMID: 31559376 Free PMC article.

2

Synthesis, biological properties and structural study of new halogenated azolo[4,5-b]pyridines as inhibitors of CK2 kinase.

Chojnacki K, Lindenblatt D, Wińska P, Wielechowska M, Toelzer C, Niefind K, Bretner M. Chojnacki K, et al. Among authors: bretner m. Bioorg Chem. 2021 Jan;106:104502. doi: 10.1016/j.bioorg.2020.104502. Epub 2020 Nov 24. Bioorg Chem. 2021. PMID: 33317841

3

Structure of the human protein kinase CK2 catalytic subunit CK2α' and interaction thermodynamics with the regulatory subunit CK2β.

Bischoff N, Olsen B, Raaf J, Bretner M, Issinger OG, Niefind K. Bischoff N, et al. Among authors: bretner m. J Mol Biol. 2011 Mar 18;407(1):1-12. doi: 10.1016/j.jmb.2011.01.020. Epub 2011 Jan 15. J Mol Biol. 2011. PMID: 21241709

4

Enzymatic activity with an incomplete catalytic spine: insights from a comparative structural analysis of human CK2α and its paralogous isoform CK2α'.

Bischoff N, Raaf J, Olsen B, Bretner M, Issinger OG, Niefind K. Bischoff N, et al. Among authors: bretner m. Mol Cell Biochem. 2011 Oct;356(1-2):57-65. doi: 10.1007/s11010-011-0948-5. Epub 2011 Jul 8. Mol Cell Biochem. 2011. PMID: 21739153

5

Biological properties and structural study of new aminoalkyl derivatives of benzimidazole and benzotriazole, dual inhibitors of CK2 and PIM1 kinases.

Chojnacki K, Wińska P, Wielechowska M, Łukowska-Chojnacka E, Tölzer C, Niefind K, Bretner M. Chojnacki K, et al. Among authors: bretner m. Bioorg Chem. 2018 Oct;80:266-275. doi: 10.1016/j.bioorg.2018.06.022. Epub 2018 Jun 22. Bioorg Chem. 2018. PMID: 29966873

6

A competition between hydrophobic and electrostatic interactions in protein-ligand systems. Binding of heterogeneously halogenated benzotriazoles by the catalytic subunit of human protein kinase CK2.

Kasperowicz S, Marzec E, Maciejewska AM, Trzybiński D, Bretner M, Woźniak K, Poznański J, Mieczkowska K. Kasperowicz S, et al. Among authors: bretner m. IUBMB Life. 2020 Jun;72(6):1211-1219. doi: 10.1002/iub.2271. Epub 2020 Mar 12. IUBMB Life. 2020. PMID: 32162783 Free article.

7

Synthesis of new analogs of benzotriazole, benzimidazole and phthalimide--potential inhibitors of human protein kinase CK2.

Najda-Bernatowicz A, Łebska M, Orzeszko A, Kopańska K, Krzywińska E, Muszyńska G, Bretner M. Najda-Bernatowicz A, et al. Among authors: bretner m. Bioorg Med Chem. 2009 Feb 15;17(4):1573-8. doi: 10.1016/j.bmc.2008.12.071. Epub 2009 Jan 7. Bioorg Med Chem. 2009. PMID: 19168362

8

Synthesis of novel polybrominated benzimidazole derivatives-potential CK2 inhibitors with anticancer and proapoptotic activity.

Łukowska-Chojnacka E, Wińska P, Wielechowska M, Poprzeczko M, Bretner M. Łukowska-Chojnacka E, et al. Among authors: bretner m. Bioorg Med Chem. 2016 Feb 15;24(4):735-41. doi: 10.1016/j.bmc.2015.12.041. Epub 2015 Dec 24. Bioorg Med Chem. 2016. PMID: 26778657

9

Synthesis of novel chiral TBBt derivatives with hydroxyl moiety. Studies on inhibition of human protein kinase CK2α and cytotoxicity properties.

Borowiecki P, Wawro AM, Wińska P, Wielechowska M, Bretner M. Borowiecki P, et al. Among authors: bretner m. Eur J Med Chem. 2014 Sep 12;84:364-74. doi: 10.1016/j.ejmech.2014.07.019. Epub 2014 Jul 11. Eur J Med Chem. 2014. PMID: 25036794

10

Synthesis, in vitro antiproliferative activity and kinase profile of new benzimidazole and benzotriazole derivatives.

Chojnacki K, Wińska P, Skierka K, Wielechowska M, Bretner M. Chojnacki K, et al. Among authors: bretner m. Bioorg Chem. 2017 Jun;72:1-10. doi: 10.1016/j.bioorg.2017.02.017. Epub 2017 Mar 16. Bioorg Chem. 2017. PMID: 28340404

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