Skip to main page content
U.S. flag

An official website of the United States government

Dot gov

The .gov means it’s official.
Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you’re on a federal government site.

Https

The site is secure.
The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.

Access keys NCBI Homepage MyNCBI Homepage Main Content Main Navigation

Search Page

Filters

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

Search Results

93 results

Filters applied: . Clear all
Results are displayed in a computed author sort order. The Results By Year timeline is not available.
Page 1
Quinoxaline derivatives as new inhibitors of coxsackievirus B5.
Carta A, Sanna G, Briguglio I, Madeddu S, Vitale G, Piras S, Corona P, Peana AT, Laurini E, Fermeglia M, Pricl S, Serra A, Carta E, Loddo R, Giliberti G. Carta A, et al. Among authors: fermeglia m. Eur J Med Chem. 2018 Feb 10;145:559-569. doi: 10.1016/j.ejmech.2017.12.083. Epub 2017 Dec 27. Eur J Med Chem. 2018. PMID: 29339251 Free article.
A combined in silico/in vitro approach unveils common molecular requirements for efficient BVDV RdRp binding of linear aromatic N-polycyclic systems.
Carta A, Briguglio I, Piras S, Corona P, Ibba R, Laurini E, Fermeglia M, Pricl S, Desideri N, Atzori EM, La Colla P, Collu G, Delogu I, Loddo R. Carta A, et al. Among authors: fermeglia m. Eur J Med Chem. 2016 Jul 19;117:321-34. doi: 10.1016/j.ejmech.2016.03.080. Epub 2016 Apr 8. Eur J Med Chem. 2016. PMID: 27161176
Pharmacophore modeling, resistant mutant isolation, docking, and MM-PBSA analysis: Combined experimental/computer-assisted approaches to identify new inhibitors of the bovine viral diarrhea virus (BVDV).
Tonelli M, Boido V, Colla P, Loddo R, Posocco P, Paneni MS, Fermeglia M, Pricl S. Tonelli M, et al. Among authors: fermeglia m. Bioorg Med Chem. 2010 Mar 15;18(6):2304-2316. doi: 10.1016/j.bmc.2010.01.058. Epub 2010 Jan 29. Bioorg Med Chem. 2010. PMID: 20189812
3-Aryl-2-[1H-benzotriazol-1-yl]acrylonitriles: a novel class of potent tubulin inhibitors.
Carta A, Briguglio I, Piras S, Boatto G, La Colla P, Loddo R, Tolomeo M, Grimaudo S, Di Cristina A, Pipitone RM, Laurini E, Paneni MS, Posocco P, Fermeglia M, Pricl S. Carta A, et al. Among authors: fermeglia m. Eur J Med Chem. 2011 Sep;46(9):4151-67. doi: 10.1016/j.ejmech.2011.06.018. Epub 2011 Jul 8. Eur J Med Chem. 2011. PMID: 21741130
Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives.
Briguglio I, Loddo R, Laurini E, Fermeglia M, Piras S, Corona P, Giunchedi P, Gavini E, Sanna G, Giliberti G, Ibba C, Farci P, La Colla P, Pricl S, Carta A. Briguglio I, et al. Among authors: fermeglia m. Eur J Med Chem. 2015 Nov 13;105:63-79. doi: 10.1016/j.ejmech.2015.10.002. Epub 2015 Oct 9. Eur J Med Chem. 2015. PMID: 26479028 Free article.
Triazolopyridinyl-acrylonitrile derivatives as antimicrotubule agents: Synthesis, in vitro and in silico characterization of antiproliferative activity, inhibition of tubulin polymerization and binding thermodynamics.
Briguglio I, Laurini E, Pirisi MA, Piras S, Corona P, Fermeglia M, Pricl S, Carta A. Briguglio I, et al. Among authors: fermeglia m. Eur J Med Chem. 2017 Dec 1;141:460-472. doi: 10.1016/j.ejmech.2017.09.065. Epub 2017 Oct 3. Eur J Med Chem. 2017. PMID: 29055869
93 results