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Discovery of furan and dihydrofuran-fused tricyclic benzo[d]imidazole derivatives as potent and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-1.
Bioorg Med Chem Lett. 2017 Dec 1;27(23):5131-5138. doi: 10.1016/j.bmcl.2017.10.062.
Bioorg Med Chem Lett. 2017.
PMID: 29100801
Synthesis and pharmacological evaluation of novel N-aryl-3,4-dihydro-1'H-spiro[chromene-2,4'-piperidine]-1'-carboxamides as TRPM8 antagonists.
Chaudhari SS, Kadam AB, Khairatkar-Joshi N, Mukhopadhyay I, Karnik PV, Raghuram A, Rao SS, Vaiyapuri TS, Wale DP, Bhosale VM, Gudi GS, Sangana RR, Thomas A.
Chaudhari SS, et al. Among authors: sangana rr.
Bioorg Med Chem. 2013 Nov 1;21(21):6542-53. doi: 10.1016/j.bmc.2013.08.031. Epub 2013 Aug 29.
Bioorg Med Chem. 2013.
PMID: 24055075
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Alleviating CYP and hERG liabilities by structure optimization of dihydrofuran-fused tricyclic benzo[d]imidazole series - Potent, selective and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-2.
Muthukaman N, Deshmukh S, Tambe M, Pisal D, Tondlekar S, Shaikh M, Sarode N, Kattige VG, Sawant P, Pisat M, Karande V, Honnegowda S, Kulkarni A, Behera D, Jadhav SB, Sangana RR, Gudi GS, Khairatkar-Joshi N, Gharat LA.
Muthukaman N, et al. Among authors: sangana rr.
Bioorg Med Chem Lett. 2018 Apr 15;28(7):1211-1218. doi: 10.1016/j.bmcl.2018.02.048. Epub 2018 Feb 28.
Bioorg Med Chem Lett. 2018.
PMID: 29519738
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Effect of Tinospora cordifolia aqua-alcoholic extract on pharmacokinetic of Glibenclamide in rat: An herb-drug interaction study.
Sahu R, Ahmed T, Sangana R, Punde R, Subudhi BB.
Sahu R, et al.
J Pharm Biomed Anal. 2018 Mar 20;151:310-316. doi: 10.1016/j.jpba.2018.01.010. Epub 2018 Jan 10.
J Pharm Biomed Anal. 2018.
PMID: 29413979
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Discovery of benzo[d]imidazo[5,1-b]thiazole as a new class of phosphodiesterase 10A inhibitors.
Banerjee A, Narayana L, Raje FA, Pisal DV, Kadam PA, Gullapalli S, Kumar H, More SV, Bajpai M, Sangana RR, Jadhav S, Gudi GS, Khairatkar-Joshi N, Merugu RR, Voleti SR, Gharat LA.
Banerjee A, et al. Among authors: sangana rr.
Bioorg Med Chem Lett. 2013 Dec 15;23(24):6747-54. doi: 10.1016/j.bmcl.2013.10.027. Epub 2013 Oct 26.
Bioorg Med Chem Lett. 2013.
PMID: 24231362
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Imidazopyridazinones as novel PDE7 inhibitors: SAR and in vivo studies in Parkinson's disease model.
Banerjee A, Patil S, Pawar MY, Gullapalli S, Gupta PK, Gandhi MN, Bhateja DK, Bajpai M, Sangana RR, Gudi GS, Khairatkar-Joshi N, Gharat LA.
Banerjee A, et al. Among authors: sangana rr.
Bioorg Med Chem Lett. 2012 Oct 1;22(19):6286-91. doi: 10.1016/j.bmcl.2012.07.077. Epub 2012 Aug 8.
Bioorg Med Chem Lett. 2012.
PMID: 22944118
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Isothiazole and isoxazole fused pyrimidones as PDE7 inhibitors: SAR and pharmacokinetic evaluation.
Banerjee A, Yadav PS, Bajpai M, Sangana RR, Gullapalli S, Gudi GS, Gharat LA.
Banerjee A, et al. Among authors: sangana rr.
Bioorg Med Chem Lett. 2012 May 1;22(9):3223-8. doi: 10.1016/j.bmcl.2012.03.025. Epub 2012 Mar 23.
Bioorg Med Chem Lett. 2012.
PMID: 22487174
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