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Anti-fibrotic Potential of AT2 Receptor Agonists.
Front Pharmacol. 2017 Aug 31;8:564. doi: 10.3389/fphar.2017.00564. eCollection 2017.
Front Pharmacol. 2017.
PMID: 28912715
Free PMC article.
Review.
Using conformational constraints at position 6 of Angiotensin II to generate compounds with enhanced AT2R selectivity and proteolytic stability.
Tourwé D, Tsiailanis AD, Parisis N, Hirmiz B, Del Borgo M, Aguilar MI, Van der Poorten O, Ballet S, Widdop RE, Tzakos AG.
Tourwé D, et al. Among authors: hirmiz b.
Bioorg Med Chem Lett. 2021 Jul 1;43:128086. doi: 10.1016/j.bmcl.2021.128086. Epub 2021 May 7.
Bioorg Med Chem Lett. 2021.
PMID: 33965531
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Single Peptide Backbone Surrogate Mutations to Regulate Angiotensin GPCR Subtype Selectivity.
Vrettos EI, Valverde IE, Mascarin A, Pallier PN, Cerofolini L, Fragai M, Parigi G, Hirmiz B, Bekas N, Grob NM, Stylos EΚ, Shaye H, Del Borgo M, Aguilar MI, Magnani F, Syed N, Crook T, Waqif E, Ghazaly E, Cherezov V, Widdop RE, Luchinat C, Michael-Titus AT, Mindt TL, Tzakos AG.
Vrettos EI, et al. Among authors: hirmiz b.
Chemistry. 2020 Aug 21;26(47):10690-10694. doi: 10.1002/chem.202000924. Epub 2020 Jul 21.
Chemistry. 2020.
PMID: 32691857
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Enhancement of glioblastoma multiforme therapy through a novel Quercetin-Losartan hybrid.
Tsiailanis AD, Renziehausen A, Kiriakidi S, Vrettos EI, Markopoulos GS, Sayyad N, Hirmiz B, Aguilar MI, Del Borgo MP, Kolettas E, Widdop RE, Mavromoustakos T, Crook T, Syed N, Tzakos AG.
Tsiailanis AD, et al. Among authors: hirmiz b.
Free Radic Biol Med. 2020 Nov 20;160:391-402. doi: 10.1016/j.freeradbiomed.2020.08.007. Epub 2020 Aug 18.
Free Radic Biol Med. 2020.
PMID: 32822744
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