Vilar S - Search Results

1

Synthesis and structure-activity relationship study of novel 3-heteroarylcoumarins based on pyridazine scaffold as selective MAO-B inhibitors.

Costas-Lago MC, Besada P, Rodríguez-Enríquez F, Viña D, Vilar S, Uriarte E, Borges F, Terán C. Costas-Lago MC, et al. Among authors: vilar s. Eur J Med Chem. 2017 Oct 20;139:1-11. doi: 10.1016/j.ejmech.2017.07.045. Epub 2017 Jul 25. Eur J Med Chem. 2017. PMID: 28797881

2

Novel (coumarin-3-yl)carbamates as selective MAO-B inhibitors: synthesis, in vitro and in vivo assays, theoretical evaluation of ADME properties and docking study.

Matos MJ, Vilar S, Gonzalez-Franco RM, Uriarte E, Santana L, Friedman C, Tatonetti NP, Viña D, Fontenla JA. Matos MJ, et al. Among authors: vilar s. Eur J Med Chem. 2013 May;63:151-61. doi: 10.1016/j.ejmech.2013.02.009. Epub 2013 Feb 16. Eur J Med Chem. 2013. PMID: 23474901

3

Synthesis, pharmacological study and docking calculations of new benzo[f]coumarin derivatives as dual inhibitors of enzymatic systems involved in neurodegenerative diseases.

Matos MJ, Janeiro P, González Franco RM, Vilar S, Tatonetti NP, Santana L, Uriarte E, Borges F, Fontenla JA, Viña D. Matos MJ, et al. Among authors: vilar s. Future Med Chem. 2014 Mar;6(4):371-83. doi: 10.4155/fmc.14.9. Future Med Chem. 2014. PMID: 24635520

4

Potent and selective MAO-B inhibitory activity: amino- versus nitro-3-arylcoumarin derivatives.

Matos MJ, Rodríguez-Enríquez F, Vilar S, Santana L, Uriarte E, Hripcsak G, Estrada M, Rodríguez-Franco MI, Viña D. Matos MJ, et al. Among authors: vilar s. Bioorg Med Chem Lett. 2015 Feb 1;25(3):642-8. doi: 10.1016/j.bmcl.2014.12.001. Epub 2014 Dec 8. Bioorg Med Chem Lett. 2015. PMID: 25532905

5

Development of novel adenosine receptor ligands based on the 3-amidocoumarin scaffold.

Matos MJ, Vilar S, Kachler S, Celeiro M, Vazquez-Rodriguez S, Santana L, Uriarte E, Hripcsak G, Borges F, Klotz KN. Matos MJ, et al. Among authors: vilar s. Bioorg Chem. 2015 Aug;61:1-6. doi: 10.1016/j.bioorg.2015.05.008. Epub 2015 May 22. Bioorg Chem. 2015. PMID: 26042529

6

New insights into highly potent tyrosinase inhibitors based on 3-heteroarylcoumarins: Anti-melanogenesis and antioxidant activities, and computational molecular modeling studies.

Pintus F, Matos MJ, Vilar S, Hripcsak G, Varela C, Uriarte E, Santana L, Borges F, Medda R, Di Petrillo A, Era B, Fais A. Pintus F, et al. Among authors: vilar s. Bioorg Med Chem. 2017 Mar 1;25(5):1687-1695. doi: 10.1016/j.bmc.2017.01.037. Epub 2017 Jan 31. Bioorg Med Chem. 2017. PMID: 28189394

7

In Silico Prediction of P-glycoprotein Binding: Insights from Molecular Docking Studies.

Vilar S, Sobarzo-Sánchez E, Uriarte E. Vilar S, et al. Curr Med Chem. 2019;26(10):1746-1760. doi: 10.2174/0929867325666171129121924. Curr Med Chem. 2019. PMID: 29189117 Review.

8

Structure-Based Optimization of Coumarin hA₃ Adenosine Receptor Antagonists.

Matos MJ, Vilar S, Vazquez-Rodriguez S, Kachler S, Klotz KN, Buccioni M, Delogu G, Santana L, Uriarte E, Borges F. Matos MJ, et al. Among authors: vilar s. J Med Chem. 2020 Mar 12;63(5):2577-2587. doi: 10.1021/acs.jmedchem.9b01572. Epub 2019 Dec 4. J Med Chem. 2020. PMID: 31738058

9

Design, synthesis, and vasorelaxant and platelet antiaggregatory activities of coumarin-resveratrol hybrids.

Vilar S, Quezada E, Santana L, Uriarte E, Yánez M, Fraiz N, Alcaide C, Cano E, Orallo F. Vilar S, et al. Bioorg Med Chem Lett. 2006 Jan 15;16(2):257-61. doi: 10.1016/j.bmcl.2005.10.013. Epub 2005 Nov 3. Bioorg Med Chem Lett. 2006. PMID: 16275073

10

Probabilistic neural network model for the in silico evaluation of anti-HIV activity and mechanism of action.

Vilar S, Santana L, Uriarte E. Vilar S, et al. J Med Chem. 2006 Feb 9;49(3):1118-24. doi: 10.1021/jm050932j. J Med Chem. 2006. PMID: 16451076

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

72 results

Search Page