Asami T - Search Results

1

Investigation of the structural requirements of K-Ras(G12D) selective inhibitory peptide KRpep-2d using alanine scans and cysteine bridging.

Niida A, Sasaki S, Yonemori K, Sameshima T, Yaguchi M, Asami T, Sakamoto K, Kamaura M. Niida A, et al. Among authors: asami t. Bioorg Med Chem Lett. 2017 Jun 15;27(12):2757-2761. doi: 10.1016/j.bmcl.2017.04.063. Epub 2017 Apr 21. Bioorg Med Chem Lett. 2017. PMID: 28457754

2

Serum stability of selected decapeptide agonists of KISS1R using pseudopeptides.

Asami T, Nishizawa N, Ishibashi Y, Nishibori K, Nakayama M, Horikoshi Y, Matsumoto S, Yamaguchi M, Matsumoto H, Tarui N, Ohtaki T, Kitada C. Asami T, et al. Bioorg Med Chem Lett. 2012 Oct 15;22(20):6391-6. doi: 10.1016/j.bmcl.2012.08.069. Epub 2012 Aug 23. Bioorg Med Chem Lett. 2012. PMID: 22975302

3

Trypsin resistance of a decapeptide KISS1R agonist containing an Nω-methylarginine substitution.

Asami T, Nishizawa N, Ishibashi Y, Nishibori K, Horikoshi Y, Matsumoto H, Ohtaki T, Kitada C. Asami T, et al. Bioorg Med Chem Lett. 2012 Oct 15;22(20):6328-32. doi: 10.1016/j.bmcl.2012.08.087. Epub 2012 Aug 30. Bioorg Med Chem Lett. 2012. PMID: 22995619

4

Design, synthesis, and biological evaluation of novel investigational nonapeptide KISS1R agonists with testosterone-suppressive activity.

Asami T, Nishizawa N, Matsui H, Nishibori K, Ishibashi Y, Horikoshi Y, Nakayama M, Matsumoto S, Tarui N, Yamaguchi M, Matsumoto H, Ohtaki T, Kitada C. Asami T, et al. J Med Chem. 2013 Nov 14;56(21):8298-307. doi: 10.1021/jm401056w. Epub 2013 Oct 17. J Med Chem. 2013. PMID: 24047141

5

Physicochemically and pharmacokinetically stable nonapeptide KISS1 receptor agonists with highly potent testosterone-suppressive activity.

Asami T, Nishizawa N, Matsui H, Takatsu Y, Suzuki A, Kiba A, Terada M, Nishibori K, Nakayama M, Ban J, Matsumoto S, Tarui N, Ikeda Y, Yamaguchi M, Kusaka M, Ohtaki T, Kitada C. Asami T, et al. J Med Chem. 2014 Jul 24;57(14):6105-15. doi: 10.1021/jm5005489. Epub 2014 Jul 7. J Med Chem. 2014. PMID: 24918545

6

Design and Synthesis of an Investigational Nonapeptide KISS1 Receptor (KISS1R) Agonist, Ac-d-Tyr-Hydroxyproline (Hyp)-Asn-Thr-Phe-azaGly-Leu-Arg(Me)-Trp-NH₂ (TAK-448), with Highly Potent Testosterone-Suppressive Activity and Excellent Water Solubility.

Nishizawa N, Takatsu Y, Kumano S, Kiba A, Ban J, Tsutsumi S, Matsui H, Matsumoto SI, Yamaguchi M, Ikeda Y, Kusaka M, Ohtaki T, Itoh F, Asami T. Nishizawa N, et al. Among authors: asami t. J Med Chem. 2016 Oct 13;59(19):8804-8811. doi: 10.1021/acs.jmedchem.6b00379. Epub 2016 Sep 21. J Med Chem. 2016. PMID: 27589480

7

Discovery of an artificial peptide agonist to the fibroblast growth factor receptor 1c/βKlotho complex from random peptide T7 phage display.

Sakamoto K, Kawata Y, Masuda Y, Umemoto T, Ito T, Asami T, Takekawa S, Ohtaki T, Inooka H. Sakamoto K, et al. Among authors: asami t. Biochem Biophys Res Commun. 2016 Nov 4;480(1):55-60. doi: 10.1016/j.bbrc.2016.10.009. Epub 2016 Oct 4. Biochem Biophys Res Commun. 2016. PMID: 27717820 Free article.

8

Novel DOCK2-selective inhibitory peptide that suppresses B-cell line migration.

Sakamoto K, Adachi Y, Komoike Y, Kamada Y, Koyama R, Fukuda Y, Kadotani A, Asami T, Sakamoto JI. Sakamoto K, et al. Among authors: asami t. Biochem Biophys Res Commun. 2017 Jan 29;483(1):183-190. doi: 10.1016/j.bbrc.2016.12.170. Epub 2016 Dec 27. Biochem Biophys Res Commun. 2017. PMID: 28039053

9

Generation of a novel artificial TrkB agonist, BM17d99, using T7 phage-displayed random peptide libraries.

Ohnishi T, Sakamoto K, Asami-Odaka A, Nakamura K, Shimizu A, Ito T, Asami T, Ohtaki T, Inooka H. Ohnishi T, et al. Among authors: asami odaka a, asami t. Biochem Biophys Res Commun. 2017 Jan 29;483(1):101-106. doi: 10.1016/j.bbrc.2016.12.186. Epub 2016 Dec 31. Biochem Biophys Res Commun. 2017. PMID: 28043792

10

Investigation on cellular uptake and pharmacodynamics of DOCK2-inhibitory peptides conjugated with cell-penetrating peptides.

Adachi Y, Sakamoto K, Umemoto T, Fukuda Y, Tani A, Asami T. Adachi Y, et al. Among authors: asami t. Bioorg Med Chem. 2017 Apr 1;25(7):2148-2155. doi: 10.1016/j.bmc.2017.02.022. Epub 2017 Feb 13. Bioorg Med Chem. 2017. PMID: 28284862

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