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Discovery of BPR1K871, a quinazoline based, multi-kinase inhibitor for the treatment of AML and solid tumors: Rational design, synthesis, in vitro and in vivo evaluation.
Hsu YC, Coumar MS, Wang WC, Shiao HY, Ke YY, Lin WH, Kuo CC, Chang CW, Kuo FM, Chen PY, Wang SY, Li AS, Chen CH, Kuo PC, Chen CP, Wu MH, Huang CL, Yen KJ, Chang YI, Hsu JT, Chen CT, Yeh TK, Song JS, Shih C, Hsieh HP. Hsu YC, et al. Among authors: huang cl. Oncotarget. 2016 Dec 27;7(52):86239-86256. doi: 10.18632/oncotarget.13369. Oncotarget. 2016. PMID: 27863392 Free PMC article.
Novel trans-2-aryl-cyclopropylamine analogues as potent and selective dipeptidyl peptidase IV inhibitors.
Tsai TY, Hsu T, Chen CT, Cheng JH, Yeh TK, Chen X, Huang CY, Chang CN, Yeh KC, Hsieh SH, Chien CH, Chang YW, Huang CH, Huang YW, Huang CL, Wu SH, Wang MH, Lu CT, Chao YS, Jiaang WT. Tsai TY, et al. Among authors: huang yw, huang cl, huang ch, huang cy. Bioorg Med Chem. 2009 Mar 15;17(6):2388-99. doi: 10.1016/j.bmc.2009.02.020. Epub 2009 Feb 20. Bioorg Med Chem. 2009. PMID: 19261480
Antitumor activities and pharmacokinetics of silatecans DB-67 and DB-91.
Yeh TK, Li CM, Chen CP, Chuu JJ, Huang CL, Wang HS, Shen CC, Lee TY, Chang CY, Chang CM, Chao YS, Lin CT, Chang JY, Chen CT. Yeh TK, et al. Among authors: huang cl. Pharmacol Res. 2010 Feb;61(2):108-15. doi: 10.1016/j.phrs.2009.07.005. Epub 2009 Jul 28. Pharmacol Res. 2010. PMID: 19643180
Intravenous paclitaxel against metastasis of human gastric tumors of diffuse type.
Tuan TF, Tsai ML, Yeh KC, Huang HC, Chung CT, Huang CL, Han CH, Chen CP, Wang MH, Shen CC, Lai YK, Lee WS, Hwang LL, Chen CT. Tuan TF, et al. Among authors: huang hc, huang cl. Cancer Chemother Pharmacol. 2010 Sep;66(4):773-83. doi: 10.1007/s00280-009-1222-3. Epub 2010 Jan 1. Cancer Chemother Pharmacol. 2010. PMID: 20044750
BPR0C261 is a novel orally active antitumor agent with antimitotic and anti-angiogenic activities.
Hu CB, Chen CP, Yeh TK, Song JS, Chang CY, Chuu JJ, Tung FF, Ho PY, Chen TW, Lin CH, Wang MH, Chang KY, Huang CL, Lin HL, Li WT, Hwang DR, Chern JH, Hwang LL, Chang JY, Chao YS, Chen CT. Hu CB, et al. Among authors: huang cl. Cancer Sci. 2011 Jan;102(1):182-91. doi: 10.1111/j.1349-7006.2010.01744.x. Epub 2010 Oct 12. Cancer Sci. 2011. PMID: 21040217 Free article.
Identification of a potent 5-phenyl-thiazol-2-ylamine-based inhibitor of FLT3 with activity against drug resistance-conferring point mutations.
Chen CT, Hsu JT, Lin WH, Lu CT, Yen SC, Hsu T, Huang YL, Song JS, Chen CH, Chou LH, Yen KJ, Chen CP, Kuo PC, Huang CL, Liu HE, Chao YS, Yeh TK, Jiaang WT. Chen CT, et al. Among authors: huang yl, huang cl. Eur J Med Chem. 2015 Jul 15;100:151-61. doi: 10.1016/j.ejmech.2015.05.008. Epub 2015 May 9. Eur J Med Chem. 2015. PMID: 26081023
Targeting Tumor Associated Phosphatidylserine with New Zinc Dipicolylamine-Based Drug Conjugates.
Liu YW, Shia KS, Wu CH, Liu KL, Yeh YC, Lo CF, Chen CT, Chen YY, Yeh TK, Chen WH, Jan JJ, Huang YC, Huang CL, Fang MY, Gray BD, Pak KY, Hsu TA, Huang KH, Tsou LK. Liu YW, et al. Among authors: huang kh, huang cl, huang yc. Bioconjug Chem. 2017 Jul 19;28(7):1878-1892. doi: 10.1021/acs.bioconjchem.7b00225. Epub 2017 Jun 19. Bioconjug Chem. 2017. PMID: 28581724
1,577 results