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Design and Synthesis of 1-((1,5-Bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)methyl)-4-methylpiperazine (BM212) and N-Adamantan-2-yl-N'-((E)-3,7-dimethylocta-2,6-dienyl)ethane-1,2-diamine (SQ109) Pyrrole Hybrid Derivatives: Discovery of Potent Antitubercular Agents Effective against Multidrug-Resistant Mycobacteria.
J Med Chem. 2016 Mar 24;59(6):2780-93. doi: 10.1021/acs.jmedchem.6b00031. Epub 2016 Mar 8.
J Med Chem. 2016.
PMID: 26907951
Free article.
Synthesis of 1,2,3-Substituted Pyrroles from Propargylamines via a One-Pot Tandem Enyne Cross Metathesis-Cyclization Reaction.
Chachignon H, Scalacci N, Petricci E, Castagnolo D.
Chachignon H, et al. Among authors: scalacci n.
J Org Chem. 2015 May 15;80(10):5287-95. doi: 10.1021/acs.joc.5b00222. Epub 2015 May 6.
J Org Chem. 2015.
PMID: 25897951
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Synthesis and SAR evaluation of novel thioridazine derivatives active against drug-resistant tuberculosis.
Scalacci N, Brown AK, Pavan FR, Ribeiro CM, Manetti F, Bhakta S, Maitra A, Smith DL, Petricci E, Castagnolo D.
Scalacci N, et al.
Eur J Med Chem. 2017 Feb 15;127:147-158. doi: 10.1016/j.ejmech.2016.12.042. Epub 2016 Dec 23.
Eur J Med Chem. 2017.
PMID: 28039773
Free article.
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Improving the Potency of N-Aryl-2,5-dimethylpyrroles against Multidrug-Resistant and Intracellular Mycobacteria.
Touitou M, Manetti F, Ribeiro CM, Pavan FR, Scalacci N, Zrebna K, Begum N, Semenya D, Gupta A, Bhakta S, McHugh TD, Senderowitz H, Kyriazi M, Castagnolo D.
Touitou M, et al. Among authors: scalacci n.
ACS Med Chem Lett. 2019 Dec 10;11(5):638-644. doi: 10.1021/acsmedchemlett.9b00515. eCollection 2020 May 14.
ACS Med Chem Lett. 2019.
PMID: 32435364
Free PMC article.
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Rethinking the old antiviral drug moroxydine: Discovery of novel analogues as anti-hepatitis C virus (HCV) agents.
Magri A, Reilly R, Scalacci N, Radi M, Hunter M, Ripoll M, Patel AH, Castagnolo D.
Magri A, et al. Among authors: scalacci n.
Bioorg Med Chem Lett. 2015 Nov 15;25(22):5372-6. doi: 10.1016/j.bmcl.2015.09.029. Epub 2015 Sep 12.
Bioorg Med Chem Lett. 2015.
PMID: 26428870
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Synthesis and Reactivity of Propargylamines in Organic Chemistry.
Lauder K, Toscani A, Scalacci N, Castagnolo D.
Lauder K, et al. Among authors: scalacci n.
Chem Rev. 2017 Dec 27;117(24):14091-14200. doi: 10.1021/acs.chemrev.7b00343. Epub 2017 Nov 22.
Chem Rev. 2017.
PMID: 29166000
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