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Arylpiperidines as a new class of oxidosqualene cyclase inhibitors.
Eur J Med Chem. 2016 Feb 15;109:13-22. doi: 10.1016/j.ejmech.2015.12.025. Epub 2015 Dec 17.
Eur J Med Chem. 2016.
PMID: 26745812
Free article.
11th German Conference on Chemoinformatics (GCC 2015) : Fulda, Germany. 8-10 November 2015.
Fechner U, de Graaf C, Torda AE, Güssregen S, Evers A, Matter H, Hessler G, Richmond NJ, Schmidtke P, Segler MHS, Waller MP, Pleik S, Shea JE, Levine Z, Mullen R, van den Broek K, Epple M, Kuhn H, Truszkowski A, Zielesny A, Fraaije JH, Gracia RS, Kast SM, Bulusu KC, Bender A, Yosipof A, Nahum O, Senderowitz H, Krotzky T, Schulz R, Wolber G, Bietz S, Rarey M, Zimmermann MO, Lange A, Ruff M, Heidrich J, Onlia I, Exner TE, Boeckler FM, Bermudez M, Firaha DS, Hollóczki O, Kirchner B, Tautermann CS, Volkamer A, Eid S, Turk S, Rippmann F, Fulle S, Saleh N, Saladino G, Gervasio FL, Haensele E, Banting L, Whitley DC, Oliveira Santos JS, Bureau R, Clark T, Sandmann A, Lanig H, Kibies P, Heil J, Hoffgaard F, Frach R, Engel J, Smith S, Basu D, Rauh D, Kohlbacher O, Boeckler FM, Essex JW, Bodnarchuk MS, Ross GA, Finkelmann AR, Göller AH, Schneider G, Husch T, Schütter C, Balducci A, Korth M, Ntie-Kang F, Günther S, Sippl W, Mbaze LM, Ntie-Kang F, Simoben CV, Lifongo LL, Ntie-Kang F, Judson P, Barilla J, Lokajíček MV, Pisaková H, Simr P, Kireeva N, Petrov A, Ostroumov D, Solovev VP, Pervov VS, Friedrich NO, Sommer K, Rarey M, Kirchmair J, Proschak E, Weber J, Moser D, Kalinowski L, Achenbach J…
See abstract for full author list ➔
Fechner U, et al. Among authors: bockler fm.
J Cheminform. 2016 Apr 26;8(Suppl 1):18. doi: 10.1186/s13321-016-0119-5.
J Cheminform. 2016.
PMID: 29270804
Free PMC article.
No abstract available.
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Data quality in drug discovery: the role of analytical performance in ligand binding assays.
Wätzig H, Oltmann-Norden I, Steinicke F, Alhazmi HA, Nachbar M, El-Hady DA, Albishri HM, Baumann K, Exner T, Böckler FM, El Deeb S.
Wätzig H, et al. Among authors: bockler fm.
J Comput Aided Mol Des. 2015 Sep;29(9):847-65. doi: 10.1007/s10822-015-9851-6. Epub 2015 Jun 13.
J Comput Aided Mol Des. 2015.
PMID: 26070362
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A highly practical RCM approach towards a molecular building kit of spirocyclic reverse turn mimics.
Bittermann H, Böckler F, Einsiedel J, Gmeiner P.
Bittermann H, et al.
Chemistry. 2006 Aug 16;12(24):6315-22. doi: 10.1002/chem.200600432.
Chemistry. 2006.
PMID: 16729342
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