Estiu G - Search Results

1

Design and synthesis of a crosslinker for studying intracellular steroid trafficking pathways.

Byrd KM, Arieno MD, Kennelly ME, Estiu G, Wiest O, Helquist P. Byrd KM, et al. Among authors: estiu g. Bioorg Med Chem. 2015 Jul 1;23(13):3843-51. doi: 10.1016/j.bmc.2015.03.053. Epub 2015 Mar 27. Bioorg Med Chem. 2015. PMID: 25890696 Free PMC article.

2

Computational studies of the cholesterol transport between NPC2 and the N-terminal domain of NPC1 (NPC1(NTD)).

Estiu G, Khatri N, Wiest O. Estiu G, et al. Biochemistry. 2013 Oct 1;52(39):6879-91. doi: 10.1021/bi4005478. Epub 2013 Sep 19. Biochemistry. 2013. PMID: 24001314

3

Identification of novel bacterial histidine biosynthesis inhibitors using docking, ensemble rescoring, and whole-cell assays.

Henriksen ST, Liu J, Estiu G, Oltvai ZN, Wiest O. Henriksen ST, et al. Among authors: estiu g. Bioorg Med Chem. 2010 Jul 15;18(14):5148-56. doi: 10.1016/j.bmc.2010.05.060. Epub 2010 Jun 1. Bioorg Med Chem. 2010. PMID: 20573514 Free PMC article.

4

Structural origin of selectivity in class II-selective histone deacetylase inhibitors.

Estiu G, Greenberg E, Harrison CB, Kwiatkowski NP, Mazitschek R, Bradner JE, Wiest O. Estiu G, et al. J Med Chem. 2008 May 22;51(10):2898-906. doi: 10.1021/jm7015254. Epub 2008 Apr 16. J Med Chem. 2008. PMID: 18412327

5

On the inhibition of histone deacetylase 8.

Estiu G, West N, Mazitschek R, Greenberg E, Bradner JE, Wiest O. Estiu G, et al. Bioorg Med Chem. 2010 Jun 1;18(11):4103-10. doi: 10.1016/j.bmc.2010.03.080. Epub 2010 Apr 3. Bioorg Med Chem. 2010. PMID: 20472442 Free PMC article.

6

Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs.

Guerra-Bubb JM, Bowers AA, Smith WB, Paranal R, Estiu G, Wiest O, Bradner JE, Williams RM. Guerra-Bubb JM, et al. Among authors: estiu g. Bioorg Med Chem Lett. 2013 Nov 1;23(21):6025-8. doi: 10.1016/j.bmcl.2013.06.012. Epub 2013 Jun 18. Bioorg Med Chem Lett. 2013. PMID: 24035339 Free PMC article.

7

Residues in the 11 A channel of histone deacetylase 1 promote catalytic activity: implications for designing isoform-selective histone deacetylase inhibitors.

Weerasinghe SV, Estiu G, Wiest O, Pflum MK. Weerasinghe SV, et al. Among authors: estiu g. J Med Chem. 2008 Sep 25;51(18):5542-51. doi: 10.1021/jm800081j. Epub 2008 Aug 27. J Med Chem. 2008. PMID: 18729444 Free PMC article.

8

Synthesis and modeling of new benzofuranone histone deacetylase inhibitors that stimulate tumor suppressor gene expression.

Charrier C, Clarhaut J, Gesson JP, Estiu G, Wiest O, Roche J, Bertrand P. Charrier C, et al. Among authors: estiu g. J Med Chem. 2009 May 14;52(9):3112-5. doi: 10.1021/jm9002439. J Med Chem. 2009. PMID: 19385600

9

Identifying ligand binding conformations of the β2-adrenergic receptor by using its agonists as computational probes.

Isin B, Estiu G, Wiest O, Oltvai ZN. Isin B, et al. Among authors: estiu g. PLoS One. 2012;7(12):e50186. doi: 10.1371/journal.pone.0050186. Epub 2012 Dec 31. PLoS One. 2012. PMID: 23300522 Free PMC article.

10

The cytoplasmic prolyl-tRNA synthetase of the malaria parasite is a dual-stage target of febrifugine and its analogs.

Herman JD, Pepper LR, Cortese JF, Estiu G, Galinsky K, Zuzarte-Luis V, Derbyshire ER, Ribacke U, Lukens AK, Santos SA, Patel V, Clish CB, Sullivan WJ Jr, Zhou H, Bopp SE, Schimmel P, Lindquist S, Clardy J, Mota MM, Keller TL, Whitman M, Wiest O, Wirth DF, Mazitschek R. Herman JD, et al. Among authors: estiu g. Sci Transl Med. 2015 May 20;7(288):288ra77. doi: 10.1126/scitranslmed.aaa3575. Sci Transl Med. 2015. PMID: 25995223 Free PMC article.

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