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Bicyclic γ-amino acids as inhibitors of γ-aminobutyrate aminotransferase.
Pinto A, Tamborini L, Pennacchietti E, Coluccia A, Silvestri R, Cullia G, De Micheli C, Conti P, De Biase D. Pinto A, et al. Among authors: cullia g. J Enzyme Inhib Med Chem. 2016;31(2):295-301. doi: 10.3109/14756366.2015.1021251. Epub 2015 Sep 25. J Enzyme Inhib Med Chem. 2016. PMID: 25807299 Free article.
Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic Activity.
Eadsforth TC, Pinto A, Luciani R, Tamborini L, Cullia G, De Micheli C, Marinelli L, Cosconati S, Novellino E, Lo Presti L, Cordeiro da Silva A, Conti P, Hunter WN, Costi MP. Eadsforth TC, et al. Among authors: cullia g. J Med Chem. 2015 Oct 22;58(20):7938-48. doi: 10.1021/acs.jmedchem.5b00687. Epub 2015 Sep 16. J Med Chem. 2015. PMID: 26322631 Free PMC article.
Folates in Trypanosoma brucei: Achievements and Opportunities.
Cullia G, Tamborini L, Conti P, De Micheli C, Pinto A. Cullia G, et al. ChemMedChem. 2018 Oct 22;13(20):2150-2158. doi: 10.1002/cmdc.201800500. Epub 2018 Sep 24. ChemMedChem. 2018. PMID: 30152195 Free article. Review.
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign.
Linciano P, Cullia G, Borsari C, Santucci M, Ferrari S, Witt G, Gul S, Kuzikov M, Ellinger B, Santarém N, Cordeiro da Silva A, Conti P, Bolognesi ML, Roberti M, Prati F, Bartoccini F, Retini M, Piersanti G, Cavalli A, Goldoni L, Bertozzi SM, Bertozzi F, Brambilla E, Rizzo V, Piomelli D, Pinto A, Bandiera T, Costi MP. Linciano P, et al. Among authors: cullia g. Eur J Med Chem. 2020 Mar 1;189:112047. doi: 10.1016/j.ejmech.2020.112047. Epub 2020 Jan 10. Eur J Med Chem. 2020. PMID: 31982652 Free article.
14 results