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Pure enantiomers of benzoylamino-tranylcypromine: LSD1 inhibition, gene modulation in human leukemia cells and effects on clonogenic potential of murine promyelocytic blasts.
Eur J Med Chem. 2015 Apr 13;94:163-74. doi: 10.1016/j.ejmech.2015.02.060. Epub 2015 Mar 3.
Eur J Med Chem. 2015.
PMID: 25768700
Structure-Reactivity Relationships on Substrates and Inhibitors of the Lysine Deacylase Sirtuin 2 from Schistosoma mansoni (SmSirt2).
Monaldi D, Rotili D, Lancelot J, Marek M, Wössner N, Lucidi A, Tomaselli D, Ramos-Morales E, Romier C, Pierce RJ, Mai A, Jung M.
Monaldi D, et al.
J Med Chem. 2019 Oct 10;62(19):8733-8759. doi: 10.1021/acs.jmedchem.9b00638. Epub 2019 Sep 20.
J Med Chem. 2019.
PMID: 31496251
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Opening the Selectivity Pocket in the Human Lysine Deacetylase Sirtuin2 - New Opportunities, New Questions.
Robaa D, Monaldi D, Wössner N, Kudo N, Rumpf T, Schiedel M, Yoshida M, Jung M.
Robaa D, et al. Among authors: monaldi d.
Chem Rec. 2018 Dec;18(12):1701-1707. doi: 10.1002/tcr.201800044. Epub 2018 Jun 21.
Chem Rec. 2018.
PMID: 29931800
Review.
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New chemical tools for probing activity and inhibition of the NAD+-dependent lysine deacylase sirtuin 2.
Swyter S, Schiedel M, Monaldi D, Szunyogh S, Lehotzky A, Rumpf T, Ovádi J, Sippl W, Jung M.
Swyter S, et al. Among authors: monaldi d.
Philos Trans R Soc Lond B Biol Sci. 2018 Jun 5;373(1748):20170083. doi: 10.1098/rstb.2017.0083.
Philos Trans R Soc Lond B Biol Sci. 2018.
PMID: 29685963
Free PMC article.
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The Statistical Style of Reasoning and the Invention of Bose-Einstein Statistics.
Monaldi D.
Monaldi D.
Ber Wiss. 2019 Dec;42(4):307-337. doi: 10.1002/bewi.201900015. Epub 2019 Dec 2.
Ber Wiss. 2019.
PMID: 31789472
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