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Multiparameter Optimization of Trypanocidal Cruzain Inhibitors With In Vivo Activity and Favorable Pharmacokinetics.
Front Pharmacol. 2022 Jan 5;12:774069. doi: 10.3389/fphar.2021.774069. eCollection 2021.
Front Pharmacol. 2022.
PMID: 35069198
Free PMC article.
Structure-Based and Molecular Modeling Studies for the Discovery of Cyclic Imides as Reversible Cruzain Inhibitors With Potent Anti-Trypanosoma cruzi Activity.
Ferreira RAA, Pauli I, Sampaio TS, de Souza ML, Ferreira LLG, Magalhães LG, Rezende CO Jr, Ferreira RS, Krogh R, Dias LC, Andricopulo AD.
Ferreira RAA, et al. Among authors: rezende co jr.
Front Chem. 2019 Nov 25;7:798. doi: 10.3389/fchem.2019.00798. eCollection 2019.
Front Chem. 2019.
PMID: 31824926
Free PMC article.
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Synthesis, structure-activity relationship and in vitro pharmacodynamics of A-ring modified caged xanthones in a preclinical model of inflammatory breast cancer.
Chantarasriwong O, Milcarek AT, Morales TH, Settle AL, Rezende CO Jr, Althufairi BD, Theodoraki MA, Alpaugh ML, Theodorakis EA.
Chantarasriwong O, et al. Among authors: rezende co jr.
Eur J Med Chem. 2019 Apr 15;168:405-413. doi: 10.1016/j.ejmech.2019.02.047. Epub 2019 Feb 20.
Eur J Med Chem. 2019.
PMID: 30831408
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Spontaneously-forming spheroids as an in vitro cancer cell model for anticancer drug screening.
Theodoraki MA, Rezende CO Jr, Chantarasriwong O, Corben AD, Theodorakis EA, Alpaugh ML.
Theodoraki MA, et al. Among authors: rezende co jr.
Oncotarget. 2015 Aug 28;6(25):21255-67. doi: 10.18632/oncotarget.4013.
Oncotarget. 2015.
PMID: 26101913
Free PMC article.
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Synthesis and Antibacterial Activity of Alkylated Diamines and Amphiphilic Amides of Quinic Acid Derivatives.
Rezende CO Jr, Oliveira LA, Oliveira BA, Almeida CG, Ferreira BS, Le Hyaric M, Carvalho GS, Lourenço MC, Batista M, Marchini FK, Silva VL, Diniz CG, Almeida MV.
Rezende CO Jr, et al.
Chem Biol Drug Des. 2015 Sep;86(3):344-50. doi: 10.1111/cbdd.12498. Epub 2015 Jan 20.
Chem Biol Drug Des. 2015.
PMID: 25528858
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Assessment of leishmanicidal and trypanocidal activities of aliphatic diamine derivatives.
Yamanaka CN, Giordani RB, Rezende CO Jr, Eger I, Kessler RL, Tonini ML, de Moraes MH, Araújo DP, Zuanazzi JA, de Almeida MV, Steindel M.
Yamanaka CN, et al. Among authors: rezende co jr.
Chem Biol Drug Des. 2013 Dec;82(6):697-704. doi: 10.1111/cbdd.12191. Epub 2013 Aug 10.
Chem Biol Drug Des. 2013.
PMID: 23865595
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