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Re-engineering of the duocarmycin structural architecture enables bioprecursor development targeting CYP1A1 and CYP2W1 for biological activity.
J Med Chem. 2013 Aug 8;56(15):6273-7. doi: 10.1021/jm4000209. Epub 2013 Jul 26.
J Med Chem. 2013.
PMID: 23844629
Free article.
Colon cancer-specific cytochrome P450 2W1 converts duocarmycin analogues into potent tumor cytotoxins.
Travica S, Pors K, Loadman PM, Shnyder SD, Johansson I, Alandas MN, Sheldrake HM, Mkrtchian S, Patterson LH, Ingelman-Sundberg M.
Travica S, et al.
Clin Cancer Res. 2013 Jun 1;19(11):2952-61. doi: 10.1158/1078-0432.CCR-13-0238. Epub 2013 Apr 15.
Clin Cancer Res. 2013.
PMID: 23589180
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CYP2W1 polymorphism: functional aspects and relation to risk for colorectal cancer.
Stenstedt K, Travica S, Guo J, Barragan I, Pors K, Patterson L, Edler D, Mkrtchian S, Johansson I, Ingelman-Sundberg M.
Stenstedt K, et al. Among authors: travica s.
Pharmacogenomics. 2013 Oct;14(13):1615-22. doi: 10.2217/pgs.13.136.
Pharmacogenomics. 2013.
PMID: 24088132
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Colorectal cancer-specific cytochrome P450 2W1: intracellular localization, glycosylation, and catalytic activity.
Gomez A, Nekvindova J, Travica S, Lee MY, Johansson I, Edler D, Mkrtchian S, Ingelman-Sundberg M.
Gomez A, et al. Among authors: travica s.
Mol Pharmacol. 2010 Dec;78(6):1004-11. doi: 10.1124/mol.110.067652. Epub 2010 Aug 30.
Mol Pharmacol. 2010.
PMID: 20805301
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[Hormone replacement therapy with 17 beta-estradiol dydrogesterone: results of a 3-month open-label study].
Grisar J, Travica S, Metka M, Pietschmann P.
Grisar J, et al. Among authors: travica s.
Wien Klin Wochenschr. 1999 Dec 23;111(24):1035-43.
Wien Klin Wochenschr. 1999.
PMID: 10677891
German.
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Clinical profile of a new hormone replacement therapy containing 2 mg 17 beta-estradiol and 10 mg dydrogesterone.
Sator MO, Nagele F, Sator P, Travica S, Gruber D, Huber JC.
Sator MO, et al. Among authors: travica s.
Maturitas. 2000 Mar 31;34(3):267-73. doi: 10.1016/s0378-5122(99)00110-3.
Maturitas. 2000.
PMID: 10717493
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