Vasu KK - Search Results

1

New insight into adenosine receptors selectivity derived from a novel series of [5-substituted-4-phenyl-1,3-thiazol-2-yl] benzamides and furamides.

Inamdar GS, Pandya AN, Thakar HM, Sudarsanam V, Kachler S, Sabbadin D, Moro S, Klotz KN, Vasu KK. Inamdar GS, et al. Among authors: vasu kk. Eur J Med Chem. 2013 May;63:924-34. doi: 10.1016/j.ejmech.2013.03.020. Epub 2013 Mar 22. Eur J Med Chem. 2013. PMID: 23685887

2

2-Amino-5-benzoyl-4-phenylthiazoles: Development of potent and selective adenosine A1 receptor antagonists.

Scheiff AB, Yerande SG, El-Tayeb A, Li W, Inamdar GS, Vasu KK, Sudarsanam V, Müller CE. Scheiff AB, et al. Among authors: vasu kk. Bioorg Med Chem. 2010 Mar 15;18(6):2195-2203. doi: 10.1016/j.bmc.2010.01.072. Epub 2010 Feb 4. Bioorg Med Chem. 2010. PMID: 20188574

3

Novel thiazole-thiophene conjugates as adenosine receptor antagonists: synthesis, biological evaluation and docking studies.

Pandya DH, Sharma JA, Jalani HB, Pandya AN, Sudarsanam V, Kachler S, Klotz KN, Vasu KK. Pandya DH, et al. Among authors: vasu kk. Bioorg Med Chem Lett. 2015 Mar 15;25(6):1306-9. doi: 10.1016/j.bmcl.2015.01.040. Epub 2015 Jan 28. Bioorg Med Chem Lett. 2015. PMID: 25686851

4

2-Amino-5-thiazolyl motif: a novel scaffold for designing anti-inflammatory agents of diverse structures.

Franklin PX, Pillai AD, Rathod PD, Yerande S, Nivsarkar M, Padh H, Vasu KK, Sudarsanam V. Franklin PX, et al. Among authors: vasu kk. Eur J Med Chem. 2008 Jan;43(1):129-34. doi: 10.1016/j.ejmech.2007.02.008. Epub 2007 Mar 1. Eur J Med Chem. 2008. PMID: 17467123

5

Pair wise binding affinity: 3D QSAR studies on a set of triazolo [1, 5-a] quinoxalines as antagonists of AMPA and KA receptors.

Sharma RN, Thakar HM, Vasu KK, Chaturvedi SC, Pancholi SS. Sharma RN, et al. Among authors: vasu kk. J Enzyme Inhib Med Chem. 2009 Aug;24(4):1008-14. doi: 10.1080/14756360802567979. J Enzyme Inhib Med Chem. 2009. PMID: 19548793

6

Design, synthesis and evaluation of novel 2-thiophen-5-yl-3H-quinazolin-4-one analogues as inhibitors of transcription factors NF-kappaB and AP-1 mediated transcriptional activation: Their possible utilization as anti-inflammatory and anti-cancer agents.

Giri RS, Thaker HM, Giordano T, Williams J, Rogers D, Vasu KK, Sudarsanam V. Giri RS, et al. Among authors: vasu kk. Bioorg Med Chem. 2010 Apr 1;18(7):2796-808. doi: 10.1016/j.bmc.2010.01.007. Epub 2010 Jan 11. Bioorg Med Chem. 2010. PMID: 20335039

7

Synthesis and evaluation of quinazolinone derivatives as inhibitors of NF-kappaB, AP-1 mediated transcription and eIF-4E mediated translational activation: inhibitors of multi-pathways involve in cancer.

Giri RS, Thaker HM, Giordano T, Chen B, Nuthalapaty S, Vasu KK, Sudarsanam V. Giri RS, et al. Among authors: vasu kk. Eur J Med Chem. 2010 Sep;45(9):3558-63. doi: 10.1016/j.ejmech.2010.04.038. Epub 2010 May 7. Eur J Med Chem. 2010. PMID: 20557982

8

Implication of novel thiazolo-thiophene derivative (MCD-KV-10) for management of asthma.

Patil D, Dash RP, Thakur SK, Pandya AN, Venkatesh P, Vasu KK, Nivsarkar M. Patil D, et al. Among authors: vasu kk. J Enzyme Inhib Med Chem. 2015 Apr;30(2):229-39. doi: 10.3109/14756366.2014.913035. Epub 2014 Jun 18. J Enzyme Inhib Med Chem. 2015. PMID: 24939098

9

Imidazo[1,2-a]pyridines linked with thiazoles/thiophene motif through keto spacer as potential cytotoxic agents and NF-κB inhibitors.

Vasu KK, Digwal CS, Pandya AN, Pandya DH, Sharma JA, Patel S, Agarwal M. Vasu KK, et al. Bioorg Med Chem Lett. 2017 Dec 15;27(24):5463-5466. doi: 10.1016/j.bmcl.2017.10.060. Epub 2017 Nov 11. Bioorg Med Chem Lett. 2017. PMID: 29138027

10

Discovery of 2-aminoimidazole and 2-amino imidazolyl-thiazoles as non-xanthine human adenosine A₃ receptor antagonists: SAR and molecular modeling studies.

Pandya AN, Baraiya AB, Jalani HB, Pandya D, Kaila JC, Kachler S, Salmaso V, Moro S, Klotz KN, Vasu KK. Pandya AN, et al. Among authors: vasu kk. Medchemcomm. 2018 Mar 13;9(4):676-684. doi: 10.1039/c7md00643h. eCollection 2018 Apr 1. Medchemcomm. 2018. PMID: 30108958 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

38 results

Search Page