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Chemical synthesis and biological validation of immobilized protein kinase inhibitory Leucettines.
Eur J Med Chem. 2013 Apr;62:728-37. doi: 10.1016/j.ejmech.2013.01.035. Epub 2013 Feb 6.
Eur J Med Chem. 2013.
PMID: 23454515
Leucettines, a class of potent inhibitors of cdc2-like kinases and dual specificity, tyrosine phosphorylation regulated kinases derived from the marine sponge leucettamine B: modulation of alternative pre-RNA splicing.
Debdab M, Carreaux F, Renault S, Soundararajan M, Fedorov O, Filippakopoulos P, Lozach O, Babault L, Tahtouh T, Baratte B, Ogawa Y, Hagiwara M, Eisenreich A, Rauch U, Knapp S, Meijer L, Bazureau JP.
Debdab M, et al. Among authors: tahtouh t.
J Med Chem. 2011 Jun 23;54(12):4172-86. doi: 10.1021/jm200274d. Epub 2011 May 26.
J Med Chem. 2011.
PMID: 21615147
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Selectivity, cocrystal structures, and neuroprotective properties of leucettines, a family of protein kinase inhibitors derived from the marine sponge alkaloid leucettamine B.
Tahtouh T, Elkins JM, Filippakopoulos P, Soundararajan M, Burgy G, Durieu E, Cochet C, Schmid RS, Lo DC, Delhommel F, Oberholzer AE, Pearl LH, Carreaux F, Bazureau JP, Knapp S, Meijer L.
Tahtouh T, et al.
J Med Chem. 2012 Nov 8;55(21):9312-30. doi: 10.1021/jm301034u. Epub 2012 Oct 8.
J Med Chem. 2012.
PMID: 22998443
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Marine-Derived 2-Aminoimidazolone Alkaloids. Leucettamine B-Related Polyandrocarpamines Inhibit Mammalian and Protozoan DYRK & CLK Kinases.
Loaëc N, Attanasio E, Villiers B, Durieu E, Tahtouh T, Cam M, Davis RA, Alencar A, Roué M, Bourguet-Kondracki ML, Proksch P, Limanton E, Guiheneuf S, Carreaux F, Bazureau JP, Klautau M, Meijer L.
Loaëc N, et al. Among authors: tahtouh t.
Mar Drugs. 2017 Oct 17;15(10):316. doi: 10.3390/md15100316.
Mar Drugs. 2017.
PMID: 29039762
Free PMC article.
Review.
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Structure-Activity Relationship in the Leucettine Family of Kinase Inhibitors.
Tahtouh T, Durieu E, Villiers B, Bruyère C, Nguyen TL, Fant X, Ahn KH, Khurana L, Deau E, Lindberg MF, Sévère E, Miege F, Roche D, Limanton E, L'Helgoual'ch JM, Burgy G, Guiheneuf S, Herault Y, Kendall DA, Carreaux F, Bazureau JP, Meijer L.
Tahtouh T, et al.
J Med Chem. 2022 Jan 27;65(2):1396-1417. doi: 10.1021/acs.jmedchem.1c01141. Epub 2021 Dec 20.
J Med Chem. 2022.
PMID: 34928152
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An AI-based novel system for predicting respiratory support in COVID-19 patients through CT imaging analysis.
Farahat IS, Sharafeldeen A, Ghazal M, Alghamdi NS, Mahmoud A, Connelly J, van Bogaert E, Zia H, Tahtouh T, Aladrousy W, Tolba AE, Elmougy S, El-Baz A.
Farahat IS, et al. Among authors: tahtouh t.
Sci Rep. 2024 Jan 8;14(1):851. doi: 10.1038/s41598-023-51053-9.
Sci Rep. 2024.
PMID: 38191606
Free PMC article.
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Genetic variation in progesterone receptor gene and ovarian cancer risk: A case control study.
Kanabekova P, Al-Awadi AM, Bauyrzhanova Z, Tahtouh T, Sarray S, Almawi WY.
Kanabekova P, et al. Among authors: tahtouh t.
Gene. 2022 Apr 30;820:146288. doi: 10.1016/j.gene.2022.146288. Epub 2022 Feb 7.
Gene. 2022.
PMID: 35143942
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LRP5 regulates the expression of STK40, a new potential target in triple-negative breast cancers.
Maubant S, Tahtouh T, Brisson A, Maire V, Némati F, Tesson B, Ye M, Rigaill G, Noizet M, Dumont A, Gentien D, Marty-Prouvost B, de Koning L, Mahmood SF, Decaudin D, Cruzalegui F, Tucker GC, Roman-Roman S, Dubois T.
Maubant S, et al. Among authors: tahtouh t.
Oncotarget. 2018 Apr 27;9(32):22586-22604. doi: 10.18632/oncotarget.25187. eCollection 2018 Apr 27.
Oncotarget. 2018.
PMID: 29854300
Free PMC article.
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