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Novel N2-substituted pyrazolo[3,4-d]pyrimidine adenosine A3 receptor antagonists: inhibition of A3-mediated human glioblastoma cell proliferation.
Taliani S, La Motta C, Mugnaini L, Simorini F, Salerno S, Marini AM, Da Settimo F, Cosconati S, Cosimelli B, Greco G, Limongelli V, Marinelli L, Novellino E, Ciampi O, Daniele S, Trincavelli ML, Martini C. Taliani S, et al. Among authors: ciampi o. J Med Chem. 2010 May 27;53(10):3954-63. doi: 10.1021/jm901785w. J Med Chem. 2010. PMID: 20408530
5-amino-2-phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one: a versatile scaffold to obtain potent and selective A3 adenosine receptor antagonists.
Da Settimo F, Primofiore G, Taliani S, Marini AM, La Motta C, Simorini F, Salerno S, Sergianni V, Tuccinardi T, Martinelli A, Cosimelli B, Greco G, Novellino E, Ciampi O, Trincavelli ML, Martini C. Da Settimo F, et al. Among authors: ciampi o. J Med Chem. 2007 Nov 15;50(23):5676-84. doi: 10.1021/jm0708376. Epub 2007 Oct 10. J Med Chem. 2007. PMID: 17927167
Substituted pyrazolo[3,4-b]pyridines as potent A1 adenosine antagonists: synthesis, biological evaluation, and development of an A1 bovine receptor model.
Tuccinardi T, Schenone S, Bondavalli F, Brullo C, Bruno O, Mosti L, Zizzari AT, Tintori C, Manetti F, Ciampi O, Trincavelli ML, Martini C, Martinelli A, Botta M. Tuccinardi T, et al. Among authors: ciampi o. ChemMedChem. 2008 Jun;3(6):898-913. doi: 10.1002/cmdc.200700355. ChemMedChem. 2008. PMID: 18338422
Mutation analysis of oxytocin gene in individuals with adult separation anxiety.
Costa B, Pini S, Martini C, Abelli M, Gabelloni P, Ciampi O, Muti M, Gesi C, Lari L, Cardini A, Mucci A, Bucci P, Lucacchini A, Cassano GB. Costa B, et al. Among authors: ciampi o. Psychiatry Res. 2009 Jul 30;168(2):87-93. doi: 10.1016/j.psychres.2008.04.009. Epub 2009 May 26. Psychiatry Res. 2009. PMID: 19473710
New 2-arylpyrazolo[3,4-c]quinoline derivatives as potent and selective human A3 adenosine receptor antagonists. Synthesis, pharmacological evaluation, and ligand-receptor modeling studies.
Colotta V, Catarzi D, Varano F, Capelli F, Lenzi O, Filacchioni G, Martini C, Trincavelli L, Ciampi O, Pugliese AM, Pedata F, Schiesaro A, Morizzo E, Moro S. Colotta V, et al. Among authors: ciampi o. J Med Chem. 2007 Aug 23;50(17):4061-74. doi: 10.1021/jm070123v. Epub 2007 Aug 1. J Med Chem. 2007. PMID: 17665891
Synthesis, ligand-receptor modeling studies and pharmacological evaluation of novel 4-modified-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-one derivatives as potent and selective human A3 adenosine receptor antagonists.
Colotta V, Catarzi D, Varano F, Lenzi O, Filacchioni G, Martini C, Trincavelli L, Ciampi O, Traini C, Pugliese AM, Pedata F, Morizzo E, Moro S. Colotta V, et al. Among authors: ciampi o. Bioorg Med Chem. 2008 Jun 1;16(11):6086-102. doi: 10.1016/j.bmc.2008.04.039. Epub 2008 Apr 24. Bioorg Med Chem. 2008. PMID: 18468446
Pyrido[2,3-e]-1,2,4-triazolo[4,3-a]pyrazin-1-one as a new scaffold to develop potent and selective human A3 adenosine receptor antagonists. Synthesis, pharmacological evaluation, and ligand-receptor modeling studies.
Colotta V, Lenzi O, Catarzi D, Varano F, Filacchioni G, Martini C, Trincavelli L, Ciampi O, Pugliese AM, Traini C, Pedata F, Morizzo E, Moro S. Colotta V, et al. Among authors: ciampi o. J Med Chem. 2009 Apr 23;52(8):2407-19. doi: 10.1021/jm8014876. J Med Chem. 2009. PMID: 19301821
22 results