Novellino E - Search Results

1

Progresses in the pursuit of aldose reductase inhibitors: the structure-based lead optimization step.

Ramunno A, Cosconati S, Sartini S, Maglio V, Angiuoli S, La Pietra V, Di Maro S, Giustiniano M, La Motta C, Da Settimo F, Marinelli L, Novellino E. Ramunno A, et al. Among authors: novellino e. Eur J Med Chem. 2012 May;51:216-26. doi: 10.1016/j.ejmech.2012.02.045. Epub 2012 Mar 5. Eur J Med Chem. 2012. PMID: 22436396

2

Novel, highly potent aldose reductase inhibitors: cyano(2-oxo-2,3-dihydroindol-3-yl)acetic acid derivatives.

Da Settimo F, Primofiore G, Da Settimo A, La Motta C, Simorini F, Novellino E, Greco G, Lavecchia A, Boldrini E. Da Settimo F, et al. Among authors: novellino e. J Med Chem. 2003 Apr 10;46(8):1419-28. doi: 10.1021/jm030762f. J Med Chem. 2003. PMID: 12672241

3

Spirohydantoin derivatives of thiopyrano[2,3-b]pyridin-4(4H)-one as potent in vitro and in vivo aldose reductase inhibitors.

Da Settimo F, Primofiore G, La Motta C, Salerno S, Novellino E, Greco G, Lavecchia A, Laneri S, Boldrini E. Da Settimo F, et al. Among authors: novellino e. Bioorg Med Chem. 2005 Jan 17;13(2):491-9. doi: 10.1016/j.bmc.2004.10.019. Bioorg Med Chem. 2005. PMID: 15598571

4

Naphtho[1,2-d]isothiazole acetic acid derivatives as a novel class of selective aldose reductase inhibitors.

Da Settimo F, Primofiore G, La Motta C, Sartini S, Taliani S, Simorini F, Marini AM, Lavecchia A, Novellino E, Boldrini E. Da Settimo F, et al. Among authors: novellino e. J Med Chem. 2005 Nov 3;48(22):6897-907. doi: 10.1021/jm050382p. J Med Chem. 2005. PMID: 16250648

5

Pyrido[1,2-a]pyrimidin-4-one derivatives as a novel class of selective aldose reductase inhibitors exhibiting antioxidant activity.

La Motta C, Sartini S, Mugnaini L, Simorini F, Taliani S, Salerno S, Marini AM, Da Settimo F, Lavecchia A, Novellino E, Cantore M, Failli P, Ciuffi M. La Motta C, et al. Among authors: novellino e. J Med Chem. 2007 Oct 4;50(20):4917-27. doi: 10.1021/jm070398a. Epub 2007 Sep 11. J Med Chem. 2007. PMID: 17845019

6

Acetic acid aldose reductase inhibitors bearing a five-membered heterocyclic core with potent topical activity in a visual impairment rat model.

La Motta C, Sartini S, Salerno S, Simorini F, Taliani S, Marini AM, Da Settimo F, Marinelli L, Limongelli V, Novellino E. La Motta C, et al. Among authors: novellino e. J Med Chem. 2008 Jun 12;51(11):3182-93. doi: 10.1021/jm701613h. Epub 2008 May 2. J Med Chem. 2008. PMID: 18452283

7

Exploiting the pyrazolo[3,4-d]pyrimidin-4-one ring system as a useful template to obtain potent adenosine deaminase inhibitors.

La Motta C, Sartini S, Mugnaini L, Salerno S, Simorini F, Taliani S, Marini AM, Da Settimo F, Lavecchia A, Novellino E, Antonioli L, Fornai M, Blandizzi C, Del Tacca M. La Motta C, et al. Among authors: novellino e. J Med Chem. 2009 Mar 26;52(6):1681-92. doi: 10.1021/jm801427r. J Med Chem. 2009. PMID: 19226143

8

Identification of anxiolytic/nonsedative agents among indol-3-ylglyoxylamides acting as functionally selective agonists at the gamma-aminobutyric acid-A (GABAA) alpha2 benzodiazepine receptor.

Taliani S, Cosimelli B, Da Settimo F, Marini AM, La Motta C, Simorini F, Salerno S, Novellino E, Greco G, Cosconati S, Marinelli L, Salvetti F, L'Abbate G, Trasciatti S, Montali M, Costa B, Martini C. Taliani S, et al. Among authors: novellino e. J Med Chem. 2009 Jun 25;52(12):3723-34. doi: 10.1021/jm9001154. J Med Chem. 2009. PMID: 19469479

9

Pursuing aldose reductase inhibitors through in situ cross-docking and similarity-based virtual screening.

Cosconati S, Marinelli L, La Motta C, Sartini S, Da Settimo F, Olson AJ, Novellino E. Cosconati S, et al. Among authors: novellino e. J Med Chem. 2009 Sep 24;52(18):5578-81. doi: 10.1021/jm901045w. J Med Chem. 2009. PMID: 19719141

10

Novel N2-substituted pyrazolo[3,4-d]pyrimidine adenosine A3 receptor antagonists: inhibition of A3-mediated human glioblastoma cell proliferation.

Taliani S, La Motta C, Mugnaini L, Simorini F, Salerno S, Marini AM, Da Settimo F, Cosconati S, Cosimelli B, Greco G, Limongelli V, Marinelli L, Novellino E, Ciampi O, Daniele S, Trincavelli ML, Martini C. Taliani S, et al. Among authors: novellino e. J Med Chem. 2010 May 27;53(10):3954-63. doi: 10.1021/jm901785w. J Med Chem. 2010. PMID: 20408530

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

740 results

Search Page