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434 results

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Page 1
New retinoid derivatives as back-ups of Adarotene.
Giannini G, Brunetti T, Battistuzzi G, Alloatti D, Quattrociocchi G, Cima MG, Merlini L, Dallavalle S, Cincinelli R, Nannei R, Vesci L, Bucci F, Foderà R, Guglielmi MB, Pisano C, Cabri W. Giannini G, et al. Bioorg Med Chem. 2012 Apr 1;20(7):2405-15. doi: 10.1016/j.bmc.2012.01.042. Epub 2012 Feb 6. Bioorg Med Chem. 2012. PMID: 22365912
A novel atypical retinoid endowed with proapoptotic and antitumor activity.
Cincinelli R, Dallavalle S, Merlini L, Penco S, Pisano C, Carminati P, Giannini G, Vesci L, Gaetano C, Illy B, Zuco V, Supino R, Zunino F. Cincinelli R, et al. Among authors: giannini g. J Med Chem. 2003 Mar 13;46(6):909-12. doi: 10.1021/jm025593y. J Med Chem. 2003. PMID: 12620066
Undersulfated and glycol-split heparins endowed with antiangiogenic activity.
Casu B, Guerrini M, Guglieri S, Naggi A, Perez M, Torri G, Cassinelli G, Ribatti D, Carminati P, Giannini G, Penco S, Pisano C, Belleri M, Rusnati M, Presta M. Casu B, et al. Among authors: giannini g. J Med Chem. 2004 Feb 12;47(4):838-48. doi: 10.1021/jm030893g. J Med Chem. 2004. PMID: 14761186
Synthesis and structure-activity relationships of a new series of retinoid-related biphenyl-4-ylacrylic acids endowed with antiproliferative and proapoptotic activity.
Cincinelli R, Dallavalle S, Nannei R, Carella S, De Zani D, Merlini L, Penco S, Garattini E, Giannini G, Pisano C, Vesci L, Carminati P, Zuco V, Zanchi C, Zunino F. Cincinelli R, et al. Among authors: giannini g. J Med Chem. 2005 Jul 28;48(15):4931-46. doi: 10.1021/jm049440h. J Med Chem. 2005. PMID: 16033272
Biological and molecular properties of a new alpha(v)beta3/alpha(v)beta5 integrin antagonist.
Belvisi L, Riccioni T, Marcellini M, Vesci L, Chiarucci I, Efrati D, Potenza D, Scolastico C, Manzoni L, Lombardo K, Stasi MA, Orlandi A, Ciucci A, Nico B, Ribatti D, Giannini G, Presta M, Carminati P, Pisano C. Belvisi L, et al. Among authors: giannini g. Mol Cancer Ther. 2005 Nov;4(11):1670-80. doi: 10.1158/1535-7163.MCT-05-0120. Mol Cancer Ther. 2005. PMID: 16275988
434 results