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Chromenones as potent bradykinin B1 antagonists.
Bioorg Med Chem Lett. 2012 Jan 1;22(1):619-22. doi: 10.1016/j.bmcl.2011.10.068. Epub 2011 Oct 28.
Bioorg Med Chem Lett. 2012.
PMID: 22088753
Discovery of dehydro-oxopiperazine acetamides as novel bradykinin B1 receptor antagonists with enhanced in vitro potency.
Qian W, Chen JJ, Human J, Aya T, Zhu J, Biswas K, Peterkin T, Hungate RW, Arik L, Johnson E, Kumar G, Joseph S, Jona J, Guo HX, Wu Z.
Qian W, et al.
Bioorg Med Chem Lett. 2012 Jan 15;22(2):1061-7. doi: 10.1016/j.bmcl.2011.11.112. Epub 2011 Dec 8.
Bioorg Med Chem Lett. 2012.
PMID: 22197141
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Discovery of novel hydroxy-thiazoles as HIF-alpha prolyl hydroxylase inhibitors: SAR, synthesis, and modeling evaluation.
Tegley CM, Viswanadhan VN, Biswas K, Frohn MJ, Peterkin TA, Chang C, Bürli RW, Dao JH, Veith H, Rogers N, Yoder SC, Biddlecome G, Tagari P, Allen JR, Hungate RW.
Tegley CM, et al. Among authors: peterkin ta.
Bioorg Med Chem Lett. 2008 Jul 15;18(14):3925-8. doi: 10.1016/j.bmcl.2008.06.031. Epub 2008 Jun 13.
Bioorg Med Chem Lett. 2008.
PMID: 18579373
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Aryl sulfones as novel bradykinin B1 receptor antagonists for treatment of chronic pain.
Biswas K, Aya T, Qian W, Peterkin TA, Chen JJ, Human J, Hungate RW, Kumar G, Arik L, Lester-Zeiner D, Biddlecome G, Manning BH, Sun H, Dong H, Huang M, Loeloff R, Johnson EJ, Askew BC.
Biswas K, et al. Among authors: peterkin ta.
Bioorg Med Chem Lett. 2008 Sep 1;18(17):4764-9. doi: 10.1016/j.bmcl.2008.07.108. Epub 2008 Jul 31.
Bioorg Med Chem Lett. 2008.
PMID: 18706809
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3-Oxo-2-piperazinyl acetamides as potent bradykinin B1 receptor antagonists for the treatment of pain and inflammation.
Chen JJ, Nguyen T, D'Amico DC, Qian W, Human J, Aya T, Biswas K, Fotsch C, Han N, Liu Q, Nishimura N, Peterkin TA, Yang K, Zhu J, Riahi BB, Hungate RW, Andersen NG, Colyer JT, Faul MM, Kamassah A, Wang J, Jona J, Kumar G, Johnson E, Askew BC.
Chen JJ, et al. Among authors: peterkin ta.
Bioorg Med Chem Lett. 2011 Jun 1;21(11):3384-9. doi: 10.1016/j.bmcl.2011.03.115. Epub 2011 Apr 7.
Bioorg Med Chem Lett. 2011.
PMID: 21514825
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Discovery of potent, orally bioavailable phthalazinone bradykinin B1 receptor antagonists.
Biswas K, Peterkin TA, Bryan MC, Arik L, Lehto SG, Sun H, Hsieh FY, Xu C, Fremeau RT, Allen JR.
Biswas K, et al. Among authors: peterkin ta.
J Med Chem. 2011 Oct 27;54(20):7232-46. doi: 10.1021/jm200808v. Epub 2011 Sep 26.
J Med Chem. 2011.
PMID: 21902230
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