Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
5 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
1,7-Disubstituted oxyindoles are potent and selective EP(3) receptor antagonists.
Bioorg Med Chem Lett. 2010 Apr 15;20(8):2658-64. doi: 10.1016/j.bmcl.2010.02.028. Epub 2010 Feb 25.
Bioorg Med Chem Lett. 2010.
PMID: 20303752
3-Acrylamide-4-aryloxyindoles: synthesis, biological evaluation and metabolic stability of potent and selective EP3 receptor antagonists.
Zhou N, Zeller W, Zhang J, Onua E, Kiselyov AS, Ramirez J, Palsdottir G, Halldorsdottir G, Andrésson T, Gurney ME, Singh J.
Zhou N, et al.
Bioorg Med Chem Lett. 2009 Mar 1;19(5):1528-31. doi: 10.1016/j.bmcl.2008.12.112. Epub 2009 Jan 8.
Bioorg Med Chem Lett. 2009.
PMID: 19188065
Item in Clipboard
Heterocyclic 1,7-disubstituted indole sulfonamides are potent and selective human EP3 receptor antagonists.
Hategan G, Polozov AM, Zeller W, Cao H, Mishra RK, Kiselyov AS, Ramirez J, Halldorsdottir G, Andrésson T, Gurney ME, Singh J.
Hategan G, et al.
Bioorg Med Chem Lett. 2009 Dec 1;19(23):6797-800. doi: 10.1016/j.bmcl.2009.09.084. Epub 2009 Sep 27.
Bioorg Med Chem Lett. 2009.
PMID: 19836233
Item in Clipboard
Discovery of novel leukotriene A4 hydrolase inhibitors based on piperidine and piperazine scaffolds.
Sandanayaka V, Mamat B, Bhagat N, Bedell L, Halldorsdottir G, Sigthorsdottir H, Andrésson T, Kiselyov A, Gurney M, Singh J.
Sandanayaka V, et al.
Bioorg Med Chem Lett. 2010 May 1;20(9):2851-4. doi: 10.1016/j.bmcl.2010.03.047. Epub 2010 Mar 12.
Bioorg Med Chem Lett. 2010.
PMID: 20371179
Item in Clipboard
Discovery of 4-[(2S)-2-{[4-(4-chlorophenoxy)phenoxy]methyl}-1-pyrrolidinyl]butanoic acid (DG-051) as a novel leukotriene A4 hydrolase inhibitor of leukotriene B4 biosynthesis.
Sandanayaka V, Mamat B, Mishra RK, Winger J, Krohn M, Zhou LM, Keyvan M, Enache L, Sullins D, Onua E, Zhang J, Halldorsdottir G, Sigthorsdottir H, Thorlaksdottir A, Sigthorsson G, Thorsteinnsdottir M, Davies DR, Stewart LJ, Zembower DE, Andresson T, Kiselyov AS, Singh J, Gurney ME.
Sandanayaka V, et al.
J Med Chem. 2010 Jan 28;53(2):573-85. doi: 10.1021/jm900838g.
J Med Chem. 2010.
PMID: 19950900
Item in Clipboard
Cite
Cite