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Fragment-based identification of Hsp90 inhibitors.
ChemMedChem. 2009 Jun;4(6):963-6. doi: 10.1002/cmdc.200900011.
ChemMedChem. 2009.
PMID: 19301319
Chiral resolution and pharmacological characterization of the enantiomers of the Hsp90 inhibitor 2-amino-7-[4-fluoro-2-(3-pyridyl)phenyl]-4-methyl-7,8-dihydro-6H-quinazolin-5-one oxime.
Amici R, Bigogno C, Boggio R, Colombo A, Courtney SM, Dal Zuffo R, Dondio G, Fusar F, Gagliardi S, Minucci S, Molteni M, Montalbetti CA, Mortoni A, Varasi M, Vultaggio S, Mercurio C.
Amici R, et al. Among authors: fusar f.
ChemMedChem. 2014 Jul;9(7):1574-85. doi: 10.1002/cmdc.201400037. Epub 2014 Apr 17.
ChemMedChem. 2014.
PMID: 24753447
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Synthesis and biological evaluation of N-hydroxyphenylacrylamides and N-hydroxypyridin-2-ylacrylamides as novel histone deacetylase inhibitors.
Thaler F, Colombo A, Mai A, Amici R, Bigogno C, Boggio R, Cappa A, Carrara S, Cataudella T, Fusar F, Gianti E, di Ventimiglia SJ, Moroni M, Munari D, Pain G, Regalia N, Sartori L, Vultaggio S, Dondio G, Gagliardi S, Minucci S, Mercurio C, Varasi M.
Thaler F, et al. Among authors: fusar f.
J Med Chem. 2010 Jan 28;53(2):822-39. doi: 10.1021/jm901502p.
J Med Chem. 2010.
PMID: 20017493
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PAT-ChIP coupled with laser microdissection allows the study of chromatin in selected cell populations from paraffin-embedded patient samples.
Amatori S, Ballarini M, Faversani A, Belloni E, Fusar F, Bosari S, Pelicci PG, Minucci S, Fanelli M.
Amatori S, et al. Among authors: fusar f.
Epigenetics Chromatin. 2014 Aug 5;7:18. doi: 10.1186/1756-8935-7-18. eCollection 2014.
Epigenetics Chromatin. 2014.
PMID: 25104973
Free PMC article.
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