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Design and synthesis of novel sulfonamide-containing bradykinin hB2 receptor antagonists. 2. Synthesis and structure-activity relationships of alpha,alpha-cycloalkylglycine sulfonamides.
J Med Chem. 2007 Feb 8;50(3):550-65. doi: 10.1021/jm061143k.
J Med Chem. 2007.
PMID: 17266207
Design and synthesis of novel sulfonamide-containing bradykinin hB2 receptor antagonists. 1. Synthesis and SAR of alpha,alpha-dimethylglycine sulfonamides.
Fattori D, Rossi C, Fincham CI, Berettoni M, Calvani F, Catrambone F, Felicetti P, Gensini M, Terracciano R, Altamura M, Bressan A, Giuliani S, Maggi CA, Meini S, Valenti C, Quartara L.
Fattori D, et al. Among authors: gensini m.
J Med Chem. 2006 Jun 15;49(12):3602-13. doi: 10.1021/jm060137l.
J Med Chem. 2006.
PMID: 16759102
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Modulation on C- and N-terminal moieties of a series of potent and selective linear tachykinin NK(2) receptor antagonists.
Gensini M, Altamura M, Dimoulas T, Fedi V, Giannotti D, Giuliani S, Guidi A, Harmat NJ, Meini S, Nannicini R, Pasqui F, Tramontana M, Triolo A, Maggi CA.
Gensini M, et al.
ChemMedChem. 2010 Jan;5(1):65-78. doi: 10.1002/cmdc.200900389.
ChemMedChem. 2010.
PMID: 19957262
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Antiproliferative and differentiating activities of a novel series of histone deacetylase inhibitors.
Binaschi M, Boldetti A, Gianni M, Maggi CA, Gensini M, Bigioni M, Parlani M, Giolitti A, Fratelli M, Valli C, Terao M, Garattini E.
Binaschi M, et al. Among authors: gensini m.
ACS Med Chem Lett. 2010 Jul 20;1(8):411-5. doi: 10.1021/ml1001163. eCollection 2010 Nov 11.
ACS Med Chem Lett. 2010.
PMID: 24900225
Free PMC article.
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Biallelic variants in CENPF causing a phenotype distinct from Strømme syndrome.
Cappuccio G, Brillante S, Tammaro R, Pinelli M, De Bernardi ML, Gensini MG, Bijlsma EK, Koopmann TT, Hoffer MJV, McDonald K, Hendon LG, Douzgou S, Deshpande C, D'Arrigo S, Torella A, Nigro V, Franco B, Brunetti-Pierri N.
Cappuccio G, et al. Among authors: gensini mg.
Am J Med Genet C Semin Med Genet. 2022 Mar;190(1):102-108. doi: 10.1002/ajmg.c.31973. Epub 2022 Apr 30.
Am J Med Genet C Semin Med Genet. 2022.
PMID: 35488810
Free PMC article.
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Reducing post-surgical adhesions utilizing a drug-enhanced device: sodium carboxymethylcellulose aqueous gel/poly(p-dioxanone) and Tranilast.
Cui H, Gensini M, Kataria R, Twaddle T, Zhang J, Wadsworth S, Petrilli J, Rodgers K, diZerega G, Cooper K.
Cui H, et al. Among authors: gensini m.
Biomed Mater. 2009 Feb;4(1):015001. doi: 10.1088/1748-6041/4/1/015001. Epub 2008 Nov 4.
Biomed Mater. 2009.
PMID: 18981543
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Cyclopropane-annelated azaoligoheterocycles by Ti-mediated intramolecular reductive cyclopropanation of cyclic amino Acid amides.
Gensini M, de Meijere A.
Gensini M, et al.
Chemistry. 2004 Feb 6;10(3):785-90. doi: 10.1002/chem.200305068.
Chemistry. 2004.
PMID: 14767944
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Stereoselective approach to hydroxyindolizidines: protection/deprotection of the nitrone functionality via cycloaddition/retrocycloaddition.
Cordero FM, Gensini M, Goti A, Brandi A.
Cordero FM, et al. Among authors: gensini m.
Org Lett. 2000 Aug 10;2(16):2475-7. doi: 10.1021/ol006125q.
Org Lett. 2000.
PMID: 10956525
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