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(2R)-2-methylchromane-2-carboxylic acids: discovery of selective PPARalpha agonists as hypolipidemic agents.
Bioorg Med Chem Lett. 2005 Jul 15;15(14):3347-51. doi: 10.1016/j.bmcl.2005.05.028.
Bioorg Med Chem Lett. 2005.
PMID: 15950464
MK-0767, a novel dual PPARalpha/gamma agonist, displays robust antihyperglycemic and hypolipidemic activities.
Doebber TW, Kelly LJ, Zhou G, Meurer R, Biswas C, Li Y, Wu MS, Ippolito MC, Chao YS, Wang PR, Wright SD, Moller DE, Berger JP.
Doebber TW, et al. Among authors: ippolito mc.
Biochem Biophys Res Commun. 2004 May 28;318(2):323-8. doi: 10.1016/j.bbrc.2004.04.032.
Biochem Biophys Res Commun. 2004.
PMID: 15120604
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(2R)-2-ethylchromane-2-carboxylic acids: discovery of novel PPARalpha/gamma dual agonists as antihyperglycemic and hypolipidemic agents.
Koyama H, Miller DJ, Boueres JK, Desai RC, Jones AB, Berger JP, MacNaul KL, Kelly LJ, Doebber TW, Wu MS, Zhou G, Wang PR, Ippolito MC, Chao YS, Agrawal AK, Franklin R, Heck JV, Wright SD, Moller DE, Sahoo SP.
Koyama H, et al. Among authors: ippolito mc.
J Med Chem. 2004 Jun 3;47(12):3255-63. doi: 10.1021/jm030621d.
J Med Chem. 2004.
PMID: 15163205
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A novel peroxisome proliferator-activated receptor alpha/gamma dual agonist demonstrates favorable effects on lipid homeostasis.
Guo Q, Sahoo SP, Wang PR, Milot DP, Ippolito MC, Wu MS, Baffic J, Biswas C, Hernandez M, Lam MH, Sharma N, Han W, Kelly LJ, MacNaul KL, Zhou G, Desai R, Heck JV, Doebber TW, Berger JP, Moller DE, Sparrow CP, Chao YS, Wright SD.
Guo Q, et al. Among authors: ippolito mc.
Endocrinology. 2004 Apr;145(4):1640-8. doi: 10.1210/en.2003-1270. Epub 2003 Dec 30.
Endocrinology. 2004.
PMID: 14701675
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High fat fed hamster, a unique animal model for treatment of diabetic dyslipidemia with peroxisome proliferator activated receptor alpha selective agonists.
Wang PR, Guo Q, Ippolito M, Wu M, Milot D, Ventre J, Doebber T, Wright SD, Chao YS.
Wang PR, et al.
Eur J Pharmacol. 2001 Sep 21;427(3):285-93. doi: 10.1016/s0014-2999(01)01249-3.
Eur J Pharmacol. 2001.
PMID: 11567659
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Regulation of lipid metabolism and gene expression by fenofibrate in hamsters.
Guo Q, Wang PR, Milot DP, Ippolito MC, Hernandez M, Burton CA, Wright SD, Chao Y.
Guo Q, et al. Among authors: ippolito mc.
Biochim Biophys Acta. 2001 Oct 31;1533(3):220-32. doi: 10.1016/s1388-1981(01)00156-1.
Biochim Biophys Acta. 2001.
PMID: 11731332
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(D)-beta-Hydroxybutyrate inhibits adipocyte lipolysis via the nicotinic acid receptor PUMA-G.
Taggart AK, Kero J, Gan X, Cai TQ, Cheng K, Ippolito M, Ren N, Kaplan R, Wu K, Wu TJ, Jin L, Liaw C, Chen R, Richman J, Connolly D, Offermanns S, Wright SD, Waters MG.
Taggart AK, et al.
J Biol Chem. 2005 Jul 22;280(29):26649-52. doi: 10.1074/jbc.C500213200. Epub 2005 Jun 1.
J Biol Chem. 2005.
PMID: 15929991
Free article.
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PPARalpha agonists reduce 11beta-hydroxysteroid dehydrogenase type 1 in the liver.
Hermanowski-Vosatka A, Gerhold D, Mundt SS, Loving VA, Lu M, Chen Y, Elbrecht A, Wu M, Doebber T, Kelly L, Milot D, Guo Q, Wang PR, Ippolito M, Chao YS, Wright SD, Thieringer R.
Hermanowski-Vosatka A, et al.
Biochem Biophys Res Commun. 2000 Dec 20;279(2):330-6. doi: 10.1006/bbrc.2000.3966.
Biochem Biophys Res Commun. 2000.
PMID: 11118287
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