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Ascorbic and 6-Br-ascorbic acid conjugates as a tool to increase the therapeutic effects of potentially central active drugs.
Eur J Pharm Sci. 2005 Mar;24(4):259-69. doi: 10.1016/j.ejps.2004.10.014. Epub 2004 Dec 19.
Eur J Pharm Sci. 2005.
PMID: 15734292
Vitamin C and 6-amino-vitamin C conjugates of diclofenac: synthesis and evaluation.
Dalpiaz A, Pavan B, Scaglianti M, Vitali F, Bortolotti F, Biondi C, Scatturin A, Manfredini S.
Dalpiaz A, et al. Among authors: scaglianti m.
Int J Pharm. 2005 Mar 3;291(1-2):171-81. doi: 10.1016/j.ijpharm.2004.07.054. Epub 2004 Dec 30.
Int J Pharm. 2005.
PMID: 15707744
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Transporter-mediated effects of diclofenamic acid and its ascorbyl pro-drug in the in vivo neurotropic activity of ascorbyl nipecotic acid conjugate.
Dalpiaz A, Pavan B, Scaglianti M, Vitali F, Bortolotti F, Biondi C, Scatturin A, Tanganelli S, Ferraro L, Prasad P, Manfredini S.
Dalpiaz A, et al. Among authors: scaglianti m.
J Pharm Sci. 2004 Jan;93(1):78-85. doi: 10.1002/jps.10532.
J Pharm Sci. 2004.
PMID: 14648638
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Design, synthesis and in vitro evaluation on HRPE cells of ascorbic and 6-bromoascorbic acid conjugates with neuroactive molecules.
Manfredini S, Vertuani S, Pavan B, Vitali F, Scaglianti M, Bortolotti F, Biondi C, Scatturin A, Prasad P, Dalpiaz A.
Manfredini S, et al. Among authors: scaglianti m.
Bioorg Med Chem. 2004 Oct 15;12(20):5453-63. doi: 10.1016/j.bmc.2004.07.043.
Bioorg Med Chem. 2004.
PMID: 15388172
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Design, synthesis and activity of ascorbic acid prodrugs of nipecotic, kynurenic and diclophenamic acids, liable to increase neurotropic activity.
Manfredini S, Pavan B, Vertuani S, Scaglianti M, Compagnone D, Biondi C, Scatturin A, Tanganelli S, Ferraro L, Prasad P, Dalpiaz A.
Manfredini S, et al. Among authors: scaglianti m.
J Med Chem. 2002 Jan 31;45(3):559-62. doi: 10.1021/jm015556r.
J Med Chem. 2002.
PMID: 11806707
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Carnitine conjugate of nipecotic acid: a new example of dual prodrug.
Napolitano C, Scaglianti M, Scalambra E, Manfredini S, Ferraro L, Beggiato S, Vertuani S.
Napolitano C, et al. Among authors: scaglianti m.
Molecules. 2009 Aug 31;14(9):3268-74. doi: 10.3390/molecules14093268.
Molecules. 2009.
PMID: 19783924
Free PMC article.
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Evaluation of steviol and its glycosides in Stevia rebaudiana leaves and commercial sweetener by ultra-high-performance liquid chromatography-mass spectrometry.
Gardana C, Scaglianti M, Simonetti P.
Gardana C, et al. Among authors: scaglianti m.
J Chromatogr A. 2010 Feb 26;1217(9):1463-70. doi: 10.1016/j.chroma.2009.12.036. Epub 2010 Jan 6.
J Chromatogr A. 2010.
PMID: 20102764
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Analysis of the polyphenolic fraction of propolis from different sources by liquid chromatography-tandem mass spectrometry.
Gardana C, Scaglianti M, Pietta P, Simonetti P.
Gardana C, et al. Among authors: scaglianti m.
J Pharm Biomed Anal. 2007 Nov 5;45(3):390-9. doi: 10.1016/j.jpba.2007.06.022. Epub 2007 Jun 30.
J Pharm Biomed Anal. 2007.
PMID: 17935924
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