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Pyrrolo[1,3]benzothiazepine-based serotonin and dopamine receptor antagonists. Molecular modeling, further structure-activity relationship studies, and identification of novel atypical antipsychotic agents.
J Med Chem. 2004 Jan 1;47(1):143-57. doi: 10.1021/jm0309811.
J Med Chem. 2004.
PMID: 14695828
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
Minetti P, Tinti MO, Carminati P, Castorina M, Di Cesare MA, Di Serio S, Gallo G, Ghirardi O, Giorgi F, Giorgi L, Piersanti G, Bartoccini F, Tarzia G.
Minetti P, et al. Among authors: di cesare ma.
J Med Chem. 2005 Nov 3;48(22):6887-96. doi: 10.1021/jm058018d.
J Med Chem. 2005.
PMID: 16250647
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Pyrrolo[1,3]benzothiazepine-based atypical antipsychotic agents. Synthesis, structure-activity relationship, molecular modeling, and biological studies.
Campiani G, Butini S, Gemma S, Nacci V, Fattorusso C, Catalanotti B, Giorgi G, Cagnotto A, Goegan M, Mennini T, Minetti P, Di Cesare MA, Mastroianni D, Scafetta N, Galletti B, Stasi MA, Castorina M, Pacifici L, Ghirardi O, Tinti O, Carminati P.
Campiani G, et al. Among authors: di cesare ma.
J Med Chem. 2002 Jan 17;45(2):344-59. doi: 10.1021/jm010982y.
J Med Chem. 2002.
PMID: 11784139
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Novel atypical antipsychotic agents: rational design, an efficient palladium-catalyzed route, and pharmacological studies.
Campiani G, Butini S, Fattorusso C, Trotta F, Gemma S, Catalanotti B, Nacci V, Fiorini I, Cagnotto A, Mereghetti I, Mennini T, Minetti P, Di Cesare MA, Stasi MA, Di Serio S, Ghirardi O, Tinti O, Carminati P.
Campiani G, et al. Among authors: di cesare ma.
J Med Chem. 2005 Mar 24;48(6):1705-8. doi: 10.1021/jm049629t.
J Med Chem. 2005.
PMID: 15771414
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ST 1535: a preferential A2A adenosine receptor antagonist.
Stasi MA, Borsini F, Varani K, Vincenzi F, Di Cesare MA, Minetti P, Ghirardi O, Carminati P.
Stasi MA, et al. Among authors: di cesare ma.
Int J Neuropsychopharmacol. 2006 Oct;9(5):575-84. doi: 10.1017/S1461145705006188. Epub 2005 Nov 23.
Int J Neuropsychopharmacol. 2006.
PMID: 16867213
Free article.
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Predictors of a response to dexmedetomidine in intubated, critically ill adult patients.
DiCesare MA, Rech MA, DeMott JM.
DiCesare MA, et al.
Pharmacotherapy. 2021 Feb;41(2):191-197. doi: 10.1002/phar.2501. Epub 2021 Feb 2.
Pharmacotherapy. 2021.
PMID: 33421200
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