3-(1H-indazol-3-ylmethyl)-1,5-benzodiazepines: CCK-A agonists that demonstrate oral activity as satiety agents

J Med Chem. 1996 Jul 5;39(14):2655-8. doi: 10.1021/jm960249k.
No abstract available

MeSH terms

  • Administration, Oral
  • Animals
  • Benzodiazepines / chemistry
  • Benzodiazepines / pharmacology*
  • Binding Sites
  • CHO Cells
  • Cholecystokinin / agonists*
  • Cricetinae
  • Gallbladder / drug effects
  • Guinea Pigs
  • Humans
  • Mice
  • Satiety Response / drug effects*
  • Structure-Activity Relationship

Substances

  • Benzodiazepines
  • Cholecystokinin