The in vivo evaluation of poly(lactic acid) microcapsules of pilocarpine hydrochloride

J Microencapsul. 1985 Oct-Dec;2(4):289-92. doi: 10.3109/02652048509033840.

Abstract

Poly(lactic acid) microcapsules of pilocarpine hydrochloride were prepared and evaluated by measuring a miotic effect in rabbits. The microcapsule suspension showed prolongation of miosis and an improved bioavailability when compared with a standard eye dosage form.

MeSH terms

  • Animals
  • Capsules
  • Female
  • Lactates
  • Lactic Acid*
  • Pilocarpine / administration & dosage*
  • Pilocarpine / pharmacology
  • Polyesters
  • Polymers
  • Pupil / drug effects
  • Rabbits

Substances

  • Capsules
  • Lactates
  • Polyesters
  • Polymers
  • Pilocarpine
  • Lactic Acid
  • poly(lactide)