Targeted Covalent Inhibitors in Drug Discovery, Chemical Biology and Beyond

Pharmaceuticals (Basel). 2024 Feb 5;17(2):206. doi: 10.3390/ph17020206.

Authors

Ricardo A M Serafim¹, Matthias Gehringer^{1

2}, Chiara Borsari³

Affiliations

¹ Department of Pharmaceutical/Medicinal Chemistry, Institute of Pharmaceutical Sciences, Eberhard Karls University Tübingen, 72076 Tübingen, Germany.
² Cluster of Excellence iFIT (EXC 2180) 'Image-Guided & Functionally Instructed Tumor Therapies', University of Tübingen, 72076 Tübingen, Germany.
³ Department of Pharmaceutical Sciences, University of Milan, 20133 Milan, Italy.

Abstract

Covalent inhibitors have experienced a revival in medicinal chemistry and chemical biology in recent decades [...].

Publication types

Editorial