Regiospecific Reduction of 4,6-Dinitrobenzimidazoles: Synthesis, Characterization, and Biological Evaluation

Chem Biodivers. 2023 Jul;20(7):e202300191. doi: 10.1002/cbdv.202300191. Epub 2023 Jun 26.

Abstract

The regiospecific reduction of 4,6-dinitrobenzimidazole derivatives leading to the corresponding 4-amino-6-nitrobenzimidazoles was studied. The identification of the formed product structures was accomplished by spectroscopic and X-ray diffraction data. The anticancer and antiparasitic activities of the synthesized compounds were examined, and promising activities against Toxoplasma gondii and Leishmania major parasites were discovered for certain 4,6-dinitrobenzimidazoles in addition to moderate anticancer activities of the 4-amino-6-nitrobenzimidazole derivatives against T. gondii cells. However, the tumor cell experiments revealed a promising sensitivity of p53-negative colon cancer cells to these compounds.

Keywords: 4,6-dinitrobenzimidazole; 4-amino-6-nitrobenzimidazoles; anticancer agents; antiparasitic agents; regiospecific reduction.

MeSH terms

  • Antiparasitic Agents / chemistry
  • Antiparasitic Agents / pharmacology
  • Leishmania major*
  • Toxoplasma*

Substances

  • Antiparasitic Agents