Phosphodiesterase-5 Inhibitory Activity of Canthin-6-One Alkaloids and the Roots of Eurycoma longifolia and Eurycoma harmandiana

Chem Biodivers. 2022 Jul;19(7):e202200121. doi: 10.1002/cbdv.202200121. Epub 2022 Jun 15.

Abstract

Eurycoma longifolia (EL) and Eurycoma harmandiana (EH) are natural medicinal plants belonging to the Simaroubaceae family, and are well-known for their ability to enhance male sexual performance. The present study investigated the phosphodiesterase-5 (PDE-5) inhibitory activity of intact roots of EL and EH. Additionally, canthin-6-one alkaloids, β-carboline alkaloids, and quassinoids were also screened for PDE-5 inhibitory activity. We developed in vitro root and callus cultures of EL and EH to determine their PDE-5 inhibitory activity. Our results indicated that canthin-6-one alkaloids, which include canthin-6-one-9-O-β-D-glucopyranoside, 9-methoxycanthin-6-one, canthin-6-one, and 9-hydroxycanthin-6-one, exhibited PDE-5 enzymatic inhibitory activity, with IC50 values of 2.86±0.23, 3.30±1.03, 4.31±0.52, and 4.66±1.13 μM, respectively. The ethanolic extract of the intact roots of EL and EH, and the in vitro root culture of EH had large amounts of canthin-6-one alkaloids (1.50±0.04, 2.12±0.03, and 3.48±0.08 mg/g dry weight, respectively), and showed potent PDE-5 inhibition. Our findings indicate that in vitro root cultures of EH may be used to replace intact plants, and canthin-6-one-9-O-β-D-glucopyranoside should be further investigated for development as a health supplement.

Keywords: Eurycoma harmandiana; Eurycoma longifolia; canthin-6-one alkaloids; erectile dysfunction; in vitro root culture; phosphodiesterase-5.

MeSH terms

  • Alkaloids* / pharmacology
  • Carbolines / pharmacology
  • Cyclic Nucleotide Phosphodiesterases, Type 5
  • Eurycoma*
  • Indole Alkaloids
  • Plant Extracts / pharmacology
  • Plant Roots

Substances

  • Alkaloids
  • Carbolines
  • Indole Alkaloids
  • Plant Extracts
  • canthin-6-one
  • Cyclic Nucleotide Phosphodiesterases, Type 5