Structural biology of kainate receptors

Neuropharmacology. 2021 Jun 1:190:108511. doi: 10.1016/j.neuropharm.2021.108511. Epub 2021 Mar 30.

Abstract

This review summarizes structural studies on kainate receptors that explain unique functional properties of this receptor family. A large number of structures have been solved for ligand binding domain dimer assemblies, giving insight into the subtype selective pharmacology of agonists, antagonists, and allosteric modulators. Structures and biochemical studies on the amino terminal domain reveal mechanisms that play a key role in assembly of heteromeric receptors. Surprisingly, structures of full length homomeric GluK2, GluK3 and heteromeric GluK2/GluK5, receptors reveal a novel structure for the desensitized state that is strikingly different from that for AMPA receptors.

Publication types

  • Research Support, N.I.H., Intramural
  • Review

MeSH terms

  • Allosteric Site
  • Animals
  • Binding Sites
  • Humans
  • Protein Multimerization
  • Protein Structure, Quaternary
  • Protein Structure, Tertiary
  • Receptors, Kainic Acid / physiology*
  • Receptors, Kainic Acid / ultrastructure
  • Structure-Activity Relationship

Substances

  • Receptors, Kainic Acid