Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic 'writers'

Epigenomics. 2020 Sep;12(17):1479-1482. doi: 10.2217/epi-2020-0203. Epub 2020 Sep 17.
No abstract available

Keywords: DNA; DNMT; HMT; SAM analogues; bisubstrate inhibitors; epigenetics; histone; methyltransferases; substrate analogues.

Publication types

  • Editorial

MeSH terms

  • DNA (Cytosine-5-)-Methyltransferase 1 / antagonists & inhibitors
  • Enzyme Inhibitors / pharmacology
  • Epigenesis, Genetic / drug effects*
  • Gene Expression Regulation / drug effects*
  • Humans

Substances

  • Enzyme Inhibitors
  • DNA (Cytosine-5-)-Methyltransferase 1