β-Turn Mimics by Chemical Ligation

Org Lett. 2020 Jun 5;22(11):4424-4428. doi: 10.1021/acs.orglett.0c01427. Epub 2020 May 14.

Abstract

We report a simple reductive amination protocol to ligate two peptides, while simultaneously installing a β-turn mimic at the ligation junction. This strategy uses commercially available materials, mild chemical conditions, and a chemoselective ligation reaction of unprotected peptide substrates accessed through standard solid phase methods. This system was implemented in a designed β-hairpin system, and biophysical analysis demonstrates effective mimicry of the β-turn.