A specific assay for JmjC domain-containing lysine demethylase and its application to inhibitor screening

Sci China Life Sci. 2019 Oct;62(10):1404-1408. doi: 10.1007/s11427-019-9582-9. Epub 2019 Sep 6.
No abstract available

MeSH terms

  • Biosensing Techniques
  • Chromatin / chemistry
  • Enzyme Inhibitors / chemistry*
  • HeLa Cells
  • High-Throughput Screening Assays
  • Humans
  • Jumonji Domain-Containing Histone Demethylases / antagonists & inhibitors*
  • Kinetics
  • Magnetic Resonance Spectroscopy
  • Methylation
  • Molecular Structure
  • NAD / chemistry
  • Protein Binding
  • Protein Conformation
  • Sensitivity and Specificity

Substances

  • Chromatin
  • Enzyme Inhibitors
  • NAD
  • Jumonji Domain-Containing Histone Demethylases